Target Details
| UniProt AC | P10636 |
|---|---|
| Gene Symbol | MAPT |
| Protein Name | Microtubule-associated protein tau |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00418 (Tubulin-binding) |
Summary
- Multi-target molecules 150
- Clinical molecules 0
- Avg pChEMBL 7.12
KEGG Pathways (4)
Associated Diseases (4)
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KBVGRKCRBVWRQG
|
9.4 | IC50 | 2 | — | |
VYVMTNNUVNSRBD
|
9.0 | Kd | 3 | — | |
UCYVFUSXGNJNEO
|
9.0 | IC50 | 2 | — | |
FIQQLONWDXAKPQ
|
8.9 | Kd | 3 | — | |
HBGNURMASUAQFL
|
8.8 | Kd | 3 | — | |
CSWYTFLVWXTIPC
|
8.8 | Kd | 3 | — | |
QLGFITMILZNZCU
|
8.8 | IC50 | 2 | — | |
QLGFITMILZNZCU
|
8.7 | IC50 | 2 | — | |
CLWLYGJCKORDAK
|
8.7 | IC50 | 2 | — | |
ITOKNBPWGKEKPE
|
8.7 | IC50 | 2 | — | |
JLPMGOFESRTFLV
|
8.7 | IC50 | 2 | — | |
PDZMLCFMZBYPNH
|
8.7 | Kd | 3 | — | |
VEZYROFGIDSNEB
|
8.7 | IC50 | 2 | — | |
KVNVGAUWCHPHOE
|
8.6 | Kd | 3 | — | |
MJIHNNLFOKEZEW
|
8.6 | Ki | 6 | — | |
NCMRFSCEYJSKBH
|
8.6 | IC50 | 2 | — | |
VWRHRENEJPEKGV
|
8.5 | IC50 | 2 | — | |
GRYSKXCHMRRJMC
|
8.3 | IC50 | 2 | — | |
UMMCMVOJRYIPSD
|
8.3 | IC50 | 2 | — | |
QCOOCCREMZWFAR
|
8.2 | IC50 | 3 | — | |
DFOUAWOLZRCIJU
|
8.1 | IC50 | 2 | — | |
MENVSADYTLLXLP
|
8.0 | IC50 | 2 | — | |
QLWFPXXGZGCHFQ
|
8.0 | IC50 | 5 | — | |
ITOKNBPWGKEKPE
|
7.9 | IC50 | 2 | — | |
KOZNFQBNKITETG
|
7.9 | IC50 | 3 | — | |
DJAGWSNSAWJXLX
|
7.8 | IC50 | 2 | — | |
FJPQYUIIAITBKJ
|
7.7 | IC50 | 2 | — | |
CJBGZDIMVHUOFK
|
7.7 | IC50 | 3 | — | |
HSDHAJSZFGKELI
|
7.6 | IC50 | 2 | — | |
QMPGWYFQWWEQDM
|
7.6 | IC50 | 2 | — | |
NXMNKSKXYYCWRN
|
7.6 | IC50 | 3 | — | |
YNDIAUKFXKEXSV
|
7.6 | Kd | 3 | — | |
OHIOZVADSRNHCG
|
7.6 | IC50 | 2 | — | |
XVNLBZLPZWXFED
|
7.6 | IC50 | 2 | — | |
YBQUWVFHSNRTQF
|
7.6 | Ki | 3 | — | |
CPNUDRZQULAFCT
|
7.6 | Ki | 3 | — | |
GIIJLYUXUBPINQ
|
7.5 | IC50 | 3 | — | |
FHAJBKJRGWQUEK
|
7.5 | IC50 | 3 | — | |
HNRLJYOIIWONBJ
|
7.5 | IC50 | 2 | — | |
OVGGMGOSCMWAHF
|
7.5 | IC50 | 2 | — | |
JRQHXUDMDHJKJZ
|
7.5 | IC50 | 2 | — | |
KZAWBYUYDLDFQY
|
7.4 | IC50 | 3 | — | |
LWBQXWADRRVTID
|
7.4 | IC50 | 2 | — | |
CKGUJEHCLFSIPS
|
7.4 | Ki | 3 | — | |
AASZBVWGEDIXLX
|
7.4 | IC50 | 2 | — | |
KVVPUEYLAZZLFF
|
7.4 | IC50 | 3 | — | |
WNHWUUHIAMMLPH
|
7.3 | IC50 | 2 | — | |
JPWPFXUIMVYLLR
|
7.3 | IC50 | 3 | — | |
PICRXLQEOXMWHZ
|
7.3 | IC50 | 3 | — | |
AOIUAVCQCDCNFO
|
7.3 | Kd | 3 | — |