Target Details
| UniProt AC | P10415 |
|---|---|
| Gene Symbol | BCL2 |
| Protein Name | Apoptosis regulator Bcl-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00452 (Bcl-2) PF02180 (BH4) |
Summary
- Multi-target molecules 1,065
- Clinical molecules 0
- Avg pChEMBL 8.33
KEGG Pathways (43)
- AGE-RAGE signaling pathway in diabetic complications
- Adrenergic signaling in cardiomyocytes
- Amyotrophic lateral sclerosis
- Apoptosis
- Apoptosis - multiple species
- Autophagy - animal
- Chemical carcinogenesis - receptor activation
- Cholinergic synapse
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Epstein-Barr virus infection
- Estrogen signaling pathway
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Gastric cancer
- HIF-1 signaling pathway
- Hedgehog signaling pathway
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- JAK-STAT signaling pathway
- Lipid and atherosclerosis
- Measles
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Neurotrophin signaling pathway
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Platinum drug resistance
- Prostate cancer
- Protein processing in endoplasmic reticulum
- Salmonella infection
- Shigellosis
- Small cell lung cancer
- Sphingolipid signaling pathway
- Toxoplasmosis
- Tuberculosis
- p53 signaling pathway
Associated Diseases (8)
Active Molecules (1,065)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OIUWBTCVUAZJAE
|
8.7 | IC50 | 2 | — | |
WZSQSANYFAMVOB
|
8.7 | IC50 | 2 | — | |
YRVPAVLYAVUTDT
|
8.7 | IC50 | 2 | — | |
BITKVXWSPCVZNM
|
8.6 | IC50 | 2 | — | |
LQBVNQSMGBZMKD
|
8.6 | IC50 | 4 | — | |
SFFPCNJXSDCYII
|
8.6 | Kd | 2 | — | |
JLSMYNRDIKMILB
|
8.6 | IC50 | 2 | — | |
GBDXIHPNFKEYMX
|
8.6 | IC50 | 2 | — | |
KNGQPRZPODEMOV
|
8.6 | IC50 | 2 | — | |
OLRQRZVJWIGRBF
|
8.6 | IC50 | 2 | — | |
WRLOQJVQFVMDGO
|
8.6 | IC50 | 2 | — | |
WTYXWIBYVCWWIB
|
8.6 | IC50 | 3 | — | |
ZGULUKQLEOFSEK
|
8.6 | IC50 | 3 | — | |
APUJKYQKFDVLIU
|
8.6 | Ki | 2 | — | |
BSTFFLGHKSOULK
|
8.6 | Ki | 2 | — | |
WTGWSMXBZCHERZ
|
8.6 | IC50 | 2 | — | |
AYDHAOVOPVDTSV
|
8.6 | Ki | 2 | — | |
AYDHAOVOPVDTSV
|
8.6 | Ki | 2 | — | |
OKGMAGAYTGWHJF
|
8.6 | IC50 | 2 | — | |
TYFBGXRJUPXWLR
|
8.6 | Ki | 2 | — | |
TYFBGXRJUPXWLR
|
8.6 | Ki | 2 | — | |
CWRACCYYXZRWBS
|
8.6 | Ki | 2 | — | |
DQHWJPZEYONOKC
|
8.6 | Ki | 2 | — | |
FJNDZQTVVZRTPL
|
8.6 | IC50 | 3 | — | |
KIQIUHGYJICHAH
|
8.6 | IC50 | 2 | — | |
CYTMJIUBRXAZBM
|
8.6 | IC50 | 2 | — | |
FSOKCGWDPWOLON
|
8.6 | IC50 | 2 | — | |
MLQIUYYDMOTIIB
|
8.6 | IC50 | 2 | — | |
CBNKESLAJNCFQS
|
8.5 | IC50 | 2 | — | |
KWVCGBRSXAGNRN
|
8.5 | Ki | 2 | — | |
BUTLNWRLMGMMFQ
|
8.5 | IC50 | 2 | — | |
HEYSOLNBDTZSGL
|
8.5 | IC50 | 2 | — | |
IFCOPXIGNKGPBZ
|
8.5 | Ki | 2 | — | |
OFDAVDOQYGEDHJ
|
8.5 | IC50 | 2 | — | |
SARKDBRGPPXLPC
|
8.5 | IC50 | 2 | — | |
DFHJXTSWBKYUPT
|
8.5 | IC50 | 2 | — | |
LIDCRGORIMWQJN
|
8.5 | IC50 | 3 | — | |
WOKKFKCBYMRFBZ
|
8.5 | Ki | 2 | — | |
NYDLJIKNIQGBPE
|
8.5 | IC50 | 2 | — | |
BMFIKSDWRTVGGF
|
8.5 | Ki | 2 | — | |
IDIQXGNUCPNJGU
|
8.5 | IC50 | 2 | — | |
QNXVCLXSDRKQNT
|
8.5 | IC50 | 2 | — | |
MLQIUYYDMOTIIB
|
8.5 | IC50 | 2 | — | |
NZMJYOLRRCMXEQ
|
8.5 | IC50 | 3 | — | |
RFNIJUHXZGDVAV
|
8.5 | IC50 | 2 | — | |
CHJRVUUHHNKMFO
|
8.5 | IC50 | 2 | — | |
XRDADZJPQLAHCT
|
8.5 | Ki | 2 | — | |
JXOFXOSSZKQKJU
|
8.5 | IC50 | 2 | — | |
UXROYCPTOCMXGY
|
8.5 | IC50 | 2 | — | |
YLMURQOFHMQRRU
|
8.5 | Ki | 2 | — |