Target Details
| UniProt AC | P10323 |
|---|---|
| Gene Symbol | ACR |
| Protein Name | Acrosin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 24
- Clinical molecules 0
- Avg pChEMBL 7.9
Associated Diseases (1)
Active Molecules (24)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NIBWPUGZCXNNPC
|
9.2 | IC50 | 2 | — | |
GXFBSLKCSCKIAZ
|
8.9 | IC50 | 2 | — | |
TYNHUYPNNVQELL
|
8.5 | IC50 | 2 | — | |
OELAPCOUDOSGBC
|
8.5 | IC50 | 2 | — | |
OZYGEJJCKTWNSX
|
8.5 | IC50 | 2 | — | |
OKURYNRXJHYADM
|
8.3 | IC50 | 2 | — | |
PXPIXLVXGYQMFM
|
8.2 | IC50 | 3 | — | |
BGWLSYXKMJTZLS
|
8.2 | IC50 | 2 | — | |
NYKHWUCIZYMQBG
|
8.1 | IC50 | 2 | — | |
VACGBZYEDFQOIU
|
8.1 | IC50 | 2 | — | |
QQEFLVAOLVLVTK
|
8.0 | IC50 | 2 | — | |
WBLXBGFONZZALG
|
7.9 | IC50 | 2 | — | |
QFHVTOHRBHBYIA
|
7.9 | IC50 | 2 | — | |
PLAZRHIWSZYQOZ
|
7.9 | IC50 | 2 | — | |
LDCRJXLYXZVDCM
|
7.8 | IC50 | 2 | — | |
AZTUARIVGDJWKF
|
7.8 | IC50 | 2 | — | |
NMSDAYXPBQAAGR
|
7.7 | IC50 | 2 | — | |
DPXQMHQTGAAOQB
|
7.6 | IC50 | 2 | — | |
QKIICUBVSHYYQV
|
7.5 | IC50 | 2 | — | |
HKVPOMHUROEOHN
|
7.5 | IC50 | 2 | — | |
PEDVWMGVIMYXMN
|
7.4 | IC50 | 2 | — | |
XEIIETAXJGZDQU
|
7.0 | IC50 | 2 | — | |
NUDMLXKJIHBMCP
|
6.5 | IC50 | 2 | — | |
SSQXQXQTZWWUDB
|
6.5 | IC50 | 2 | — |