Target Details
| UniProt AC | P10275 |
|---|---|
| Gene Symbol | AR |
| Protein Name | Androgen receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02166 (Androgen_recep) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 364
- Clinical molecules 37
- Avg pChEMBL 6.87
KEGG Pathways (4)
Associated Diseases (5)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLZXITGNUVWIEP
|
6.8 | Ki | 2 | — | |
RJAYIUMTPVLORX
|
6.8 | IC50 | 2 | — | |
QWPDENUMNMUTHR
|
6.8 | IC50 | 2 | — | |
MWIXIWILHMYRGD
|
6.8 | IC50 | 3 | — | |
PDXCFTVMFXAKMC
|
6.8 | Ki | 2 | — | |
UZNBZDTUBTWOBU
|
6.8 | Ki | 4 | — | |
MKXKFYHWDHIYRV
|
6.8 | IC50 | 2 | — | |
ACDLPCXLODOBHE
|
6.8 | IC50 | 3 | — | |
NLPNUYHHRWOSGM
|
6.8 | IC50 | 4 | — | |
RRWMFEXUNNLRMV
|
6.8 | IC50 | 2 | — | |
BNYATMGZJPIGMW
|
6.8 | IC50 | 2 | — | |
DOGQPEOXOGREDU
|
6.8 | IC50 | 2 | — | |
HZJNRURPDVTSAA
|
6.8 | IC50 | 4 | Yes | |
HZJNRURPDVTSAA
|
6.8 | IC50 | 4 | Yes | |
WGGMBWMYJSVPSG
|
6.8 | IC50 | 3 | — | |
DFZYMRBKXQWSTE
|
6.8 | IC50 | 3 | — | |
PHKKCWVLOCDAJQ
|
6.8 | IC50 | 4 | Yes | |
NTCBYBDADUSXSB
|
6.8 | IC50 | 9 | Yes | |
RTYKMFMHRRYCIK
|
6.7 | Ki | 2 | — | |
WVCKFHDLPYAJOU
|
6.7 | IC50 | 5 | — | |
KIOOLNRTWPFVHX
|
6.7 | IC50 | 2 | — | |
CJZROCCAPJVVQO
|
6.7 | IC50 | 3 | — | |
LKJPYSCBVHEWIU
|
6.7 | IC50 | 2 | — | |
YDRMSDHDYRAUBR
|
6.7 | IC50 | 2 | — | |
MEFYNCWNNHNHMN
|
6.7 | IC50 | 3 | — | |
RVMQWZWBBBUEFH
|
6.7 | Ki | 2 | — | |
JHVKBJJTUMIPIT
|
6.7 | IC50 | 5 | — | |
POQODJWQWWICOY
|
6.7 | IC50 | 2 | — | |
PRCXSDHAGJJCKC
|
6.7 | IC50 | 2 | — | |
QLCLQHCJXWSVTF
|
6.7 | IC50 | 3 | — | |
QADHLRWLCPCEKT
|
6.7 | IC50 | 5 | Yes | |
WZKWYTSJJZVJLU
|
6.7 | IC50 | 3 | — | |
MIAURGNSNSBTNK
|
6.7 | Ki | 4 | — | |
HLAUTXJGHQLNRA
|
6.6 | IC50 | 2 | — | |
KPKCYUMBFMYREG
|
6.6 | Ki | 3 | — | |
QADHLRWLCPCEKT
|
6.6 | IC50 | 4 | — | |
WDXRGPWQVHZTQJ
|
6.6 | IC50 | 5 | — | |
MFAGIEMFDDDLMT
|
6.6 | Ki | 3 | — | |
CPUIRDMVUBPAPK
|
6.6 | Ki | 3 | — | |
PHIKAOOZNGLKDI
|
6.6 | Ki | 4 | — | |
QWPDOAPBJDUXDW
|
6.6 | IC50 | 2 | — | |
UHRXKJFPPKYYEC
|
6.6 | IC50 | 2 | — | |
MPFVEJCVRPLSQN
|
6.6 | IC50 | 2 | — | |
YTFZTDYRARTMPD
|
6.6 | IC50 | 2 | — | |
ZWTCGJWGJMGWIM
|
6.6 | Ki | 3 | — | |
HMOAZJHSXXENHE
|
6.6 | IC50 | 3 | — | |
HMOAZJHSXXENHE
|
6.6 | IC50 | 3 | — | |
NGNZPJWDMRRGGD
|
6.6 | IC50 | 2 | — | |
RUBRWONSGNOQIS
|
6.6 | IC50 | 2 | — | |
UBRFDZVHGGUVEL
|
6.6 | IC50 | 2 | — |