Target Details
| UniProt AC | P10275 |
|---|---|
| Gene Symbol | AR |
| Protein Name | Androgen receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02166 (Androgen_recep) PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 364
- Clinical molecules 37
- Avg pChEMBL 6.87
KEGG Pathways (4)
Associated Diseases (5)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IZUMHFDUSAWWQU
|
10.0 | IC50 | 2 | — | |
PUQSDJZESAQGQS
|
9.7 | IC50 | 2 | — | |
PDMMFKSKQVNJMI
|
9.6 | Ki | 2 | — | |
HGHRCZOIYJBGPL
|
9.5 | IC50 | 2 | — | |
CXFSVKGROITHRY
|
9.2 | Ki | 3 | — | |
RJZJEPYCJHLWQR
|
9.2 | IC50 | 2 | — | |
CCCIJQPRIXGQOE
|
9.1 | Kd | 4 | — | |
FVNZFSAGJPHSHT
|
9.0 | IC50 | 2 | — | |
XCAOBUOTWGIJFB
|
9.0 | IC50 | 2 | — | |
XFVHCXVBLVMUSO
|
9.0 | IC50 | 2 | — | |
AHBGXQDJONQGOL
|
8.7 | IC50 | 2 | — | |
CXFSVKGROITHRY
|
8.7 | Ki | 2 | — | |
HGHRCZOIYJBGPL
|
8.7 | IC50 | 3 | — | |
NRQQDFFSJPVQFQ
|
8.7 | IC50 | 2 | — | |
NVKAWKQGWWIWPM
|
8.7 | Ki | 5 | — | |
YMBWIGXCZKHYQH
|
8.6 | Ki | 2 | — | |
PSGAAPLEWMOORI
|
8.5 | Ki | 11 | Yes | |
QUJQBNBSMHJFAG
|
8.5 | IC50 | 2 | — | |
YXFRGFFRCABTFT
|
8.4 | Ki | 2 | — | |
MUMGGOZAMZWBJJ
|
8.4 | IC50 | 6 | — | |
AECUUHUGTSTYSJ
|
8.3 | Ki | 2 | — | |
VTRALRXIBUAIMP
|
8.3 | IC50 | 2 | — | |
KAVBXXNJZQGZIT
|
8.2 | IC50 | 2 | — | |
LGTLOCBNEXITRB
|
8.2 | Ki | 4 | — | |
GKQWMOXIBZCMDJ
|
8.2 | IC50 | 3 | — | |
FPFITAPEARIFHY
|
8.2 | IC50 | 2 | — | |
GTZWEKOQKQIWQD
|
8.2 | IC50 | 2 | — | |
XMBUPPIEVAFYHO
|
8.2 | Ki | 2 | — | |
DZKSHTKHHHLSGZ
|
8.1 | IC50 | 3 | — | |
GJMNAFGEUJBOCE
|
8.1 | IC50 | 5 | Yes | |
QIMSMVYRWNZWBL
|
8.1 | IC50 | 2 | — | |
QIMSMVYRWNZWBL
|
8.1 | IC50 | 2 | — | |
UDMCMALCRGIISA
|
8.1 | IC50 | 2 | — | |
ZDCMJDVSSLHLLQ
|
8.1 | Ki | 9 | Yes | |
UFZZMZCIWOEUKP
|
8.0 | Ki | 4 | — | |
HEVNCDKNAJNJPY
|
8.0 | Ki | 2 | — | |
QNHUAOAFGVCXEA
|
8.0 | IC50 | 4 | Yes | |
RJKFOVLPORLFTN
|
7.9 | Ki | 10 | Yes | |
ARBYGDBJECGMGA
|
7.8 | IC50 | 2 | — | |
GUVXCWSUCSDGOW
|
7.8 | IC50 | 2 | — | |
LRQSPCAZHXKTHC
|
7.8 | Ki | 3 | — | |
MBZGPEHCTCTXRE
|
7.7 | Ki | 2 | — | |
UHIOHBCVVQJMBM
|
7.7 | Ki | 2 | — | |
UWFYSQMTEOIJJG
|
7.7 | IC50 | 3 | — | |
MCZDFWOPLACFDA
|
7.7 | IC50 | 2 | — | |
VOXZDWNPVJITMN
|
7.7 | IC50 | 8 | — | |
REWRFXZVVOUSFK
|
7.7 | IC50 | 2 | — | |
DLXBCJBMEVKPIX
|
7.7 | Ki | 9 | Yes | |
XEJSGXDGPYBWNF
|
7.7 | Ki | 2 | — | |
UWFYSQMTEOIJJG
|
7.7 | IC50 | 2 | — |