Target Details
| UniProt AC | P10253 |
|---|---|
| Gene Symbol | GAA |
| Protein Name | Lysosomal alpha-glucosidase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13802 (Gal_mutarotas_2) PF01055 (Glyco_hydro_31_2nd) PF21365 (Glyco_hydro_31_3rd) PF00088 (Trefoil) |
Summary
- Multi-target molecules 93
- Clinical molecules 0
- Avg pChEMBL 6.78
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UQRORFVVSGFNRO
|
7.0 | IC50 | 3 | — | |
WKRFFFKQZNAJPZ
|
6.9 | IC50 | 4 | — | |
KRNOSIJCJVCXKU
|
6.9 | Ki | 2 | — | |
AAKDPDFZMNYDLR
|
6.8 | Ki | 3 | — | |
UMLRUQZDVOCKFS
|
6.8 | IC50 | 4 | — | |
KYZJSQCMASBHFW
|
6.7 | IC50 | 4 | — | |
HCZQIIVHWYFIPW
|
6.7 | Ki | 2 | — | |
YSPOPRLBQLNQLB
|
6.5 | IC50 | 4 | — | |
CLVUFWXGNIFGNC
|
6.5 | IC50 | 2 | — | |
CJVYZIYCASBJMV
|
6.4 | IC50 | 4 | — | |
CXYOUYJDHKEEAA
|
6.4 | IC50 | 4 | — | |
DBUBVKHVPSNEOS
|
6.4 | IC50 | 4 | — | |
KSIVPSATVMHIHN
|
6.4 | IC50 | 4 | — | |
LXDOEDROAAJZEC
|
6.4 | IC50 | 4 | — | |
MXMGYHCULWEFBE
|
6.4 | IC50 | 4 | — | |
QATMYEQOERZLRT
|
6.4 | IC50 | 4 | — | |
QHOZUKAWJGYOPU
|
6.4 | IC50 | 4 | — | |
QWUROZLZLLJOJB
|
6.4 | IC50 | 4 | — | |
SFPZLYYGRQAWHP
|
6.4 | IC50 | 4 | — | |
VDZWEGFPUVKNDZ
|
6.4 | IC50 | 4 | — | |
XVYLNHVEAOOEGI
|
6.4 | IC50 | 5 | — | |
YVSLGGVBTXNUDN
|
6.4 | IC50 | 4 | — | |
YYQBRGMRDBWZCK
|
6.4 | IC50 | 4 | — | |
ZDXDJNIBDUSCNF
|
6.4 | IC50 | 4 | — | |
XUFXOAAUWZOOIT
|
6.4 | Ki | 5 | — | |
ISOXQDJRTFFLOQ
|
6.3 | IC50 | 4 | — | |
XVYLNHVEAOOEGI
|
6.3 | IC50 | 4 | — | |
LRBVOQKEZQPBGV
|
6.3 | IC50 | 4 | — | |
ZOBPZXTWZATXDG
|
6.3 | IC50 | 4 | — | |
CTZVSPAIQWVNDN
|
6.3 | IC50 | 4 | — | |
GBWDKSXWTQIOKT
|
6.3 | IC50 | 4 | — | |
GCSIYCPYAWNIJF
|
6.3 | IC50 | 4 | — | |
HIBYDAIXVMHDLP
|
6.3 | IC50 | 4 | — | |
OLOMJUAIHOQTRI
|
6.3 | IC50 | 4 | — | |
QAEHYTHSLYSVMY
|
6.3 | IC50 | 4 | — | |
RAZNKKMSLYQFAQ
|
6.3 | IC50 | 4 | — | |
YAZFVSUANGBNBJ
|
6.3 | IC50 | 4 | — | |
ZHIDWEDSQDSXBK
|
6.3 | IC50 | 5 | — | |
IBAQFPQHRJAVAV
|
6.2 | IC50 | 3 | — | |
DSKHTMGMKRQCTC
|
6.2 | IC50 | 4 | — | |
IIHXPVAHXKBRBL
|
6.2 | IC50 | 2 | — | |
IDYFPAYNMJRQRG
|
6.2 | IC50 | 4 | — | |
AHYWGPQILWVHMI
|
6.0 | Ki | 2 | — |