Target Details
| UniProt AC | P10253 |
|---|---|
| Gene Symbol | GAA |
| Protein Name | Lysosomal alpha-glucosidase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13802 (Gal_mutarotas_2) PF01055 (Glyco_hydro_31_2nd) PF21365 (Glyco_hydro_31_3rd) PF00088 (Trefoil) |
Summary
- Multi-target molecules 93
- Clinical molecules 0
- Avg pChEMBL 6.78
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (93)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDWIUZGUDGQYDS
|
7.4 | IC50 | 4 | — | |
AMDWOVGTJFDXNB
|
7.2 | IC50 | 4 | — | |
BKWHEXSGYMNKFI
|
7.2 | IC50 | 4 | — | |
BQXPUDCETZOLFA
|
7.2 | IC50 | 4 | — | |
BQZYCKWBULGLCM
|
7.2 | IC50 | 4 | — | |
CLMLAHFQGFQGBH
|
7.2 | IC50 | 4 | — | |
CMKYOZFHMOYFFW
|
7.2 | IC50 | 4 | — | |
DFQMLPROAMKZHV
|
7.2 | IC50 | 4 | — | |
DJFRLDMXHCKQIE
|
7.2 | IC50 | 4 | — | |
FBMKVCYXVOPCAM
|
7.2 | IC50 | 4 | — | |
FZDXUZYVIOHODE
|
7.2 | IC50 | 4 | — | |
KJKCLWYPWNFEIR
|
7.2 | IC50 | 4 | — | |
LEGPWFRXOZKOPB
|
7.2 | IC50 | 4 | — | |
LLSMPIIORNDHQT
|
7.2 | IC50 | 4 | — | |
LUWIINFHVAGLPY
|
7.2 | IC50 | 4 | — | |
NHRVZBQDFATMFT
|
7.2 | IC50 | 4 | — | |
OGNSINLRDPYSFZ
|
7.2 | IC50 | 4 | — | |
OSXNVRYFODBDNK
|
7.2 | IC50 | 4 | — | |
PXWADJFLOZBBAZ
|
7.2 | IC50 | 4 | — | |
RJSPFQQBNIPXHF
|
7.2 | IC50 | 4 | — | |
SSAKKINTGKXOKU
|
7.2 | IC50 | 4 | — | |
VNCCWNPEVKBQLL
|
7.2 | IC50 | 4 | — | |
WAOPKWQPMNKXGV
|
7.2 | IC50 | 4 | — | |
YKUVPZUHOIVVDU
|
7.2 | IC50 | 4 | — | |
YTNFAKBVUZHUDI
|
7.2 | IC50 | 4 | — | |
ZLMXTRYWTKXSAV
|
7.2 | IC50 | 4 | — | |
UMTQAFJDZIIIII
|
7.1 | IC50 | 4 | — | |
ARAYTLMMNFVZHR
|
7.0 | IC50 | 4 | — | |
BLDCCWFGEGBZCI
|
7.0 | IC50 | 4 | — | |
DOVNOCXCCHSCHG
|
7.0 | IC50 | 4 | — | |
DQPWZPUYWABSPF
|
7.0 | IC50 | 4 | — | |
DRPQWESDZCGEOR
|
7.0 | IC50 | 4 | — | |
IGQHPEVZMXGBBU
|
7.0 | IC50 | 4 | — | |
PJYJNEZKIXYQCC
|
7.0 | IC50 | 4 | — | |
SAPWTKCQKHRZRO
|
7.0 | IC50 | 4 | — | |
UUUWGBCDINHYFO
|
7.0 | IC50 | 4 | — | |
YKGZMYUUPAKENG
|
7.0 | IC50 | 4 | — | |
ZEYCMWHOPSVRDV
|
7.0 | IC50 | 4 | — | |
LXBIFEVIBLOUGU
|
7.0 | IC50 | 5 | — | |
MBQCNYZEYQQTEE
|
7.0 | Ki | 2 | — | |
BMQPJEJYTZAMHH
|
7.0 | IC50 | 4 | — | |
BNTKAWOVIFJCCP
|
7.0 | IC50 | 4 | — | |
KNEYMTFGIXGZSH
|
7.0 | IC50 | 4 | — | |
NDKDJTJPQZFXFS
|
7.0 | IC50 | 4 | — | |
NPNAVSNQFQXKRQ
|
7.0 | IC50 | 4 | — | |
PPISPTPDBFRCBK
|
7.0 | IC50 | 4 | — | |
PUJSLUAPZZYXAC
|
7.0 | IC50 | 4 | — | |
RLZJJGBOXWUGPZ
|
7.0 | IC50 | 4 | — | |
SCXRCOCVOIVRLD
|
7.0 | IC50 | 4 | — | |
ULKUTHGPRZMYRV
|
7.0 | IC50 | 4 | — |