Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CYEUKAQPQWGZPP
|
6.1 | IC50 | 2 | — | |
QAGJBUHXUXXXNX
|
6.1 | IC50 | 2 | — | |
VFTACXMSOLUDDR
|
6.1 | IC50 | 2 | — | |
AICFZQPLVSSSFU
|
6.1 | IC50 | 2 | — | |
RZGWXIMFXSAXRM
|
6.1 | IC50 | 4 | — | |
QBIWXGCBGBHXON
|
6.1 | IC50 | 2 | — | |
CTJDSJGCDMNHRC
|
6.1 | Kd | 2 | — | |
GEXHQXMZXYXJPR
|
6.1 | Kd | 2 | — | |
JTEAXQGGYNNSDQ
|
6.1 | IC50 | 2 | — | |
KIYZRANEFPEAJE
|
6.1 | IC50 | 2 | — | |
QEKGJLUOEDTRIW
|
6.1 | IC50 | 2 | — | |
QIXFKLPOAIIFGF
|
6.1 | IC50 | 2 | — | |
YIEPOGUSSKXXSP
|
6.1 | IC50 | 2 | — | |
CFQSYTCHYSNACR
|
6.1 | IC50 | 2 | — | |
DFVOOMGEUDYSTE
|
6.1 | IC50 | 2 | — | |
ORKNIPZHPCWIDI
|
6.1 | IC50 | 2 | — | |
QSAYMUXKFGQYQN
|
6.1 | IC50 | 2 | — | |
SHSPLTGUTOVZEW
|
6.1 | IC50 | 2 | — | |
YGALISXJEIZOHZ
|
6.1 | IC50 | 2 | — | |
HOCBJBNQIQQQGT
|
6.1 | IC50 | 10 | — | |
IIRZRWSQPNYQNC
|
6.1 | IC50 | 2 | — | |
KEHDYFXOYPSDFQ
|
6.1 | Ki | 3 | — | |
LIENCHBZNNMNKG
|
6.1 | IC50 | 2 | — | |
WBLZKCOFIDSWKH
|
6.1 | Kd | 2 | — | |
GGPZRFLFVXMBEZ
|
6.1 | IC50 | 2 | — | |
ACGUYXCXAPNIKK
|
6.0 | IC50 | 11 | Yes | |
KPPRBOLFVPVWMS
|
6.0 | IC50 | 2 | — | |
NENXLTIJMAMZOM
|
6.0 | IC50 | 2 | — | |
MJJALKDDGIKVBE
|
6.0 | IC50 | 30 | Yes | |
WVXFUFQTNVWHME
|
6.0 | IC50 | 2 | — | |
LHBIUOYHJIXRST
|
6.0 | IC50 | 2 | — | |
RZTKCADKVFEBSP
|
6.0 | IC50 | 2 | — | |
FMYKJLXRRQTBOR
|
6.0 | IC50 | 3 | — | |
IQVFCZXMGASAGI
|
6.0 | IC50 | 2 | — | |
RJWLAIMXRBDUMH
|
6.0 | IC50 | 2 | — | |
JRHFOWQWUVMCHX
|
6.0 | Ki | 5 | — | |
XCUCLKWBHWYCEZ
|
6.0 | IC50 | 2 | — |