Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRNGPDUFHQXSOZ
|
6.3 | IC50 | 2 | — | |
LSFMSEYLICBQLD
|
6.3 | IC50 | 2 | — | |
LSFMSEYLICBQLD
|
6.3 | IC50 | 2 | — | |
LVLPBPSLLDDHMK
|
6.3 | IC50 | 2 | — | |
MMOGDCKWHZFLMO
|
6.3 | IC50 | 2 | — | |
MRSXETXDOITHNK
|
6.3 | IC50 | 2 | — | |
MVMXSHQQBNAWMC
|
6.3 | IC50 | 2 | — | |
OYEOCKYUCQUKMH
|
6.3 | IC50 | 2 | — | |
OYEOCKYUCQUKMH
|
6.3 | IC50 | 2 | — | |
QFWWLRCXQIIMLA
|
6.3 | IC50 | 2 | — | |
QJDMARSQHXLLBE
|
6.3 | IC50 | 2 | — | |
RCFGNCPIHMGBGF
|
6.3 | IC50 | 2 | — | |
RFISFJYBBQQZPY
|
6.3 | IC50 | 2 | — | |
RUJRCMWJRKOZTO
|
6.3 | IC50 | 2 | — | |
SIQVSLICJZAZGM
|
6.3 | IC50 | 2 | — | |
UEGSTNJPMSGHMF
|
6.3 | IC50 | 2 | — | |
VQJHSXBJTLPKHO
|
6.3 | IC50 | 2 | — | |
VVXBKZFYMWTAHG
|
6.3 | IC50 | 2 | — | |
VYYDFJQUXALHPF
|
6.3 | IC50 | 2 | — | |
VYYDFJQUXALHPF
|
6.3 | IC50 | 2 | — | |
XHWLSZIPRUJMBX
|
6.3 | IC50 | 2 | — | |
XHWLSZIPRUJMBX
|
6.3 | IC50 | 2 | — | |
YCSCOAGMDRJISW
|
6.3 | IC50 | 2 | — | |
ZSSDZVMVWPPHTJ
|
6.3 | IC50 | 2 | — | |
ZZNLHLJRATZLSO
|
6.3 | IC50 | 2 | — | |
DGZUMJXQUNLVNS
|
6.2 | IC50 | 2 | — | |
NJXPUSRCRCOWEQ
|
6.2 | IC50 | 2 | — | |
DBRXOUCRJQVYJQ
|
6.2 | IC50 | 4 | — | |
JSASWRWALCMOQP
|
6.2 | IC50 | 2 | — | |
UKTOBRQSOYSYJK
|
6.2 | IC50 | 2 | — | |
FMPUADOXTPMTON
|
6.2 | IC50 | 2 | — | |
QLWOSILDDBBNKU
|
6.2 | Ki | 2 | — | |
UTDZHTFBLCBKHG
|
6.2 | IC50 | 2 | — | |
JZRRCGQQCZGHEA
|
6.2 | IC50 | 2 | — | |
JPWOPFCHHBSUKB
|
6.2 | IC50 | 4 | — | |
JAZGKZKQQSCVMM
|
6.2 | IC50 | 2 | — | |
NDXWDWBHDSNJNP
|
6.2 | IC50 | 2 | — | |
NFWQGKLIEDRSFG
|
6.2 | IC50 | 2 | — | |
YPCBLSVBUXIGNW
|
6.2 | IC50 | 2 | — | |
RYGJIKURQDMMQZ
|
6.2 | IC50 | 2 | — | |
DYEFUKCXAQOFHX
|
6.2 | IC50 | 31 | — | |
FSWBAMMIGFKJBV
|
6.2 | IC50 | 6 | — | |
MEWSAFKJOGMCKZ
|
6.2 | IC50 | 2 | — | |
NLVRHQFXQFSBQK
|
6.2 | IC50 | 2 | — | |
CMRWLYLCXJHAMP
|
6.2 | IC50 | 2 | — | |
MKZYMKKUBVPEET
|
6.2 | Ki | 2 | — | |
NDXWDWBHDSNJNP
|
6.2 | IC50 | 2 | — | |
RXNNWOBJWBKPHT
|
6.2 | IC50 | 2 | — | |
AXRYRYVKAWYZBR
|
6.2 | Ki | 6 | — | |
UGSXTJOTPOFHOD
|
6.2 | IC50 | 2 | — |