Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPUBNLAIJOZWSC
|
6.6 | IC50 | 2 | — | |
VGAAKAWUEJYBSO
|
6.6 | IC50 | 2 | — | |
VOZFVBDEURHNMJ
|
6.6 | IC50 | 2 | — | |
WDJUZGPOPHTGOT
|
6.6 | IC50 | 11 | — | |
APIGQOKYEQLSCD
|
6.6 | IC50 | 2 | — | |
HWBPESUHQMIXLB
|
6.6 | IC50 | 2 | — | |
LUMXDKZMUPIRHM
|
6.6 | IC50 | 2 | — | |
HKNJCUVSQUGVHP
|
6.6 | IC50 | 2 | — | |
BQHNOSUNTGCFNQ
|
6.6 | IC50 | 2 | — | |
CHRXGLBKPPPZDY
|
6.6 | IC50 | 2 | — | |
IGVYCVBUHQMNRZ
|
6.6 | IC50 | 2 | — | |
MTDXSRBZZFMIHM
|
6.6 | IC50 | 2 | — | |
ZSDMEQDHYASRTO
|
6.6 | IC50 | 2 | — | |
FIAFUQMPZJWCLV
|
6.6 | IC50 | 9 | — | |
JVLIBXIZJUCZPD
|
6.6 | IC50 | 2 | — | |
MQVYGJYJHLBMAT
|
6.6 | IC50 | 2 | — | |
LMXOHSDXUQEUSF
|
6.6 | IC50 | 6 | — | |
LERCEIGOROJLAY
|
6.5 | IC50 | 2 | — | |
LQCVZCCEYLDBQM
|
6.5 | IC50 | 2 | — | |
PUDFTLRNHLQJHN
|
6.5 | IC50 | 2 | — | |
RJMUSRYZPJIFPJ
|
6.5 | IC50 | 3 | — | |
UDXIYOCRUKPXES
|
6.5 | IC50 | 2 | — | |
VCQYBHSDNWQLAS
|
6.5 | IC50 | 2 | — | |
WDMSWWUPIMEGNZ
|
6.5 | IC50 | 2 | — | |
PLMXOHHVTRBRNY
|
6.5 | IC50 | 2 | — | |
CLVRPAZDBOBROH
|
6.5 | IC50 | 2 | — | |
PMJIHLSCWIDGMD
|
6.5 | IC50 | 4 | — | |
QBPGYDYJTIUYEC
|
6.5 | IC50 | 2 | — | |
ONHLDSBQCBVYJW
|
6.5 | IC50 | 2 | — | |
VGSWJDSJKKUBMQ
|
6.5 | IC50 | 2 | — | |
ITFVOMQMGITEDI
|
6.5 | IC50 | 2 | — | |
BMGLKHIACFLVAZ
|
6.5 | IC50 | 2 | — | |
JZRRCGQQCZGHEA
|
6.5 | IC50 | 2 | — | |
KRXMYBAZKJBJAB
|
6.5 | IC50 | 2 | — | |
XAAUOSGFCRLDMO
|
6.5 | IC50 | 2 | — | |
NAOYSRBUEYWQNL
|
6.4 | IC50 | 3 | — | |
ZPEDAVGOVRCNQR
|
6.4 | IC50 | 2 | — | |
XOTUFJPCITWJHW
|
6.4 | IC50 | 2 | — | |
ZZRPDKZPYYZHPR
|
6.4 | IC50 | 2 | — | |
AUZONCFQVSMFAP
|
6.4 | IC50 | 15 | — | |
HRFSFFXXTXEMAV
|
6.4 | IC50 | 2 | — | |
BOJLJKMUGYYKCZ
|
6.4 | IC50 | 2 | — | |
MJIHNNLFOKEZEW
|
6.4 | IC50 | 6 | — | |
PKMUHQIDVVOXHQ
|
6.4 | IC50 | 2 | — | |
QYENXTYKACLCGO
|
6.4 | IC50 | 2 | — | |
PHUZMTSQHVZDOX
|
6.4 | IC50 | 2 | — | |
RCEGRHOAYJTPPY
|
6.4 | IC50 | 2 | — | |
ZSVNOTCVAYHYOM
|
6.4 | IC50 | 2 | — | |
GWBBUNQDUSRZEQ
|
6.4 | IC50 | 2 | — | |
HZTJOSBNLNQPCX
|
6.4 | IC50 | 2 | — |