Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUEGVRNFVNRCFT
|
7.0 | IC50 | 2 | — | |
IGVYCVBUHQMNRZ
|
7.0 | IC50 | 2 | — | |
OTSRIQAQJQPBAR
|
6.9 | IC50 | 2 | — | |
GHBWVWMKFOCWLG
|
6.9 | IC50 | 2 | — | |
GJCBTWHGKCNYAB
|
6.9 | IC50 | 2 | — | |
MXEYFHLZFXXVGA
|
6.9 | IC50 | 2 | — | |
DVCCOMHGZJHYKJ
|
6.9 | Ki | 2 | — | |
KDMQSUUXKLZVNU
|
6.9 | IC50 | 4 | — | |
JHNYAIWXEJSBGF
|
6.9 | IC50 | 2 | — | |
JDSJDASOXWCHPN
|
6.8 | IC50 | 2 | — | |
KFGXONJZGIXSGH
|
6.8 | IC50 | 2 | — | |
ODVBBZFQPGORMJ
|
6.8 | IC50 | 2 | — | |
IGUWUTUJRGNIDR
|
6.8 | IC50 | 2 | — | |
KEGCOZYNPKOENI
|
6.8 | IC50 | 2 | — | |
PVXINZLXDUDSLJ
|
6.8 | IC50 | 2 | — | |
VZIYPNWVVYEAOU
|
6.8 | IC50 | 2 | — | |
IZEKFCXSFNUWAM
|
6.8 | IC50 | 19 | — | |
AFZSMODLJJCVPP
|
6.8 | IC50 | 12 | — | |
LILMGDHNUAKBHW
|
6.8 | IC50 | 2 | — | |
WQYWUTMBHBBLCS
|
6.8 | IC50 | 2 | — | |
WUKOFKVFVKFOQQ
|
6.8 | IC50 | 2 | — | |
AKZKTNZCQWEVFQ
|
6.8 | IC50 | 2 | — | |
IGVYCVBUHQMNRZ
|
6.8 | IC50 | 2 | — | |
QHXIEOUYOSYVEB
|
6.8 | IC50 | 2 | — | |
UIXRRGFIAVPQEF
|
6.8 | IC50 | 2 | — | |
WBJZVUPGWANLHC
|
6.8 | IC50 | 3 | — | |
WKNCKKOHQQLNCY
|
6.8 | IC50 | 3 | — | |
YHMHUCMMFCCPCT
|
6.8 | IC50 | 2 | — | |
UJNIZUGKDDYPEP
|
6.8 | IC50 | 2 | — | |
OYXVEGKFFGZMOT
|
6.8 | IC50 | 2 | — | |
CFHDKPIYROJEMW
|
6.7 | Ki | 2 | — | |
QUIIIYITNGOFEI
|
6.7 | IC50 | 3 | — | |
LTMHDMANZUZIPE
|
6.7 | IC50 | 10 | — | |
QOJHUOHZVTVTCS
|
6.7 | IC50 | 2 | — | |
RDZZBPHZWCRITM
|
6.7 | IC50 | 3 | — | |
SFEJHJONVMMWHN
|
6.7 | IC50 | 2 | — | |
UOCKRIUAKQUEKQ
|
6.7 | IC50 | 2 | — | |
YTTSOCJNZAYJTJ
|
6.7 | Ki | 2 | — | |
CWAHMAWZJYIHRF
|
6.7 | IC50 | 2 | — | |
FOLCUFKJHSQMEL
|
6.7 | IC50 | 3 | — | |
NFQUTFRPWQDRIQ
|
6.7 | IC50 | 2 | — | |
IGVYCVBUHQMNRZ
|
6.7 | IC50 | 2 | — | |
JGRJVKVZQYCAHT
|
6.7 | IC50 | 2 | — | |
NLGZYIOUBQCYSZ
|
6.7 | IC50 | 2 | — | |
MRORARXZMFZSPG
|
6.7 | IC50 | 2 | — | |
NAQVFTHUFHJOPN
|
6.7 | IC50 | 2 | — | |
ZJUKTBDSGOFHSH
|
6.7 | IC50 | 22 | — | |
NELMAQCQYVSAFW
|
6.7 | IC50 | 3 | — | |
UKSIDTWNLGQRED
|
6.7 | IC50 | 2 | — | |
BLRXSZOWSREMKN
|
6.6 | IC50 | 2 | — |