Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LJTINUKMKJKLBT
|
7.4 | IC50 | 2 | — | |
ZYTJDBYJYAWQKF
|
7.4 | IC50 | 3 | — | |
GMRHLFCOAHOGTL
|
7.4 | IC50 | 2 | — | |
GACCXUQYGGYVOX
|
7.4 | IC50 | 2 | — | |
VGULVEAJHVXHOO
|
7.4 | IC50 | 2 | — | |
CKIKEFAXGVRFNU
|
7.3 | Ki | 2 | — | |
NSMKRGLMOMZSEI
|
7.3 | IC50 | 2 | — | |
URRVDEBIADJRJN
|
7.3 | IC50 | 2 | — | |
FGVVTMRZYROCTH
|
7.3 | IC50 | 2 | Yes | |
KUAZQDVKQLNFPE
|
7.3 | IC50 | 9 | — | |
XXWDDQJFYNJUCB
|
7.3 | IC50 | 3 | — | |
BHQBUUBHCKLKLD
|
7.3 | IC50 | 2 | — | |
CZFNHMDDLQKLAQ
|
7.3 | IC50 | 2 | — | |
HPKJGHVHQWJOOT
|
7.3 | IC50 | 2 | — | |
HPKJGHVHQWJOOT
|
7.3 | IC50 | 2 | — | |
ZMOZSXJGWLKEFR
|
7.3 | IC50 | 2 | — | |
WSVWWSLUPXQXHY
|
7.3 | IC50 | 2 | — | |
YVCYGQVRUNWVOI
|
7.3 | IC50 | 3 | — | |
RJLLYBLMSBFMNO
|
7.3 | IC50 | 2 | — | |
UXGYVCSOFAFCGA
|
7.2 | Ki | 2 | — | |
QCRLRBSKQJIUTG
|
7.2 | IC50 | 3 | — | |
UINAKWUAROHCQN
|
7.2 | Ki | 2 | — | |
WGQKYBSKWIADBV
|
7.2 | IC50 | 2 | — | |
LZINVNIRRCILMQ
|
7.2 | IC50 | 2 | — | |
NSUKAWKDBSYLPB
|
7.2 | IC50 | 2 | — | |
JXGIYKRRPGCLFV
|
7.2 | Ki | 2 | — | |
NFQUTFRPWQDRIQ
|
7.2 | IC50 | 2 | — | |
GQTHPXZAMKDSPN
|
7.1 | IC50 | 2 | — | |
ZTDJZRYPBSMEET
|
7.1 | IC50 | 2 | — | |
PYOUAIQXJALPKW
|
7.1 | IC50 | 2 | — | |
ZBWCAPBPHSAJFD
|
7.1 | IC50 | 2 | — | |
GTBAQTKMASRCMG
|
7.1 | IC50 | 2 | — | |
IBMWPTXMJVFLFJ
|
7.1 | IC50 | 2 | — | |
PAVJYVVZIJTAHT
|
7.1 | IC50 | 2 | — | |
GELYEKCYUJJOCW
|
7.1 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
7.1 | IC50 | 7 | — | |
CVJBJRQQYWUAPJ
|
7.1 | IC50 | 2 | — | |
GDKLDALGJZVEKT
|
7.1 | IC50 | 2 | — | |
QOTVXHVQJYHEFL
|
7.1 | IC50 | 2 | — | |
XCUAIINAJCDIPM
|
7.0 | IC50 | 2 | — | |
ICJGURDUFOHBQH
|
7.0 | Ki | 2 | — | |
IIYSOKUNCMQEPQ
|
7.0 | IC50 | 2 | — | |
JNJYSDKMQGAPIR
|
7.0 | IC50 | 2 | — | |
INCPOQCTPBWLJW
|
7.0 | IC50 | 2 | — | |
QCHRRORBILDLMB
|
7.0 | IC50 | 2 | — | |
YFUZVOLEKQFVCQ
|
7.0 | IC50 | 3 | — | |
MTXAPYGDANDQKT
|
7.0 | IC50 | 2 | — | |
QGNQEKJDMJPWOT
|
7.0 | IC50 | 2 | — | |
RCEIITLUVHPUBP
|
7.0 | IC50 | 2 | — | |
CUEGVRNFVNRCFT
|
7.0 | IC50 | 2 | — |