Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HROGANPCJBTDFB
|
8.0 | IC50 | 2 | — | |
UAFLFCJAOKBHAW
|
8.0 | IC50 | 2 | — | |
UOAJBSPQDBHHRC
|
8.0 | IC50 | 2 | — | |
ZMUQNKRTLPRFGB
|
8.0 | IC50 | 2 | — | |
QJCAWERZKXLFIJ
|
7.9 | IC50 | 2 | — | |
YUUOVSLHZXGIKO
|
7.9 | IC50 | 2 | — | |
FTIFIZZEWIBTMR
|
7.8 | IC50 | 2 | — | |
IYZRWOMTSMYRCM
|
7.8 | Ki | 2 | — | |
CJDAPCDGESTEPR
|
7.8 | IC50 | 4 | — | |
KOUVVHAGIUSYCU
|
7.8 | IC50 | 2 | — | |
KTAAIKREGSDHNS
|
7.8 | IC50 | 4 | — | |
QMOLFHLCHURCHA
|
7.8 | IC50 | 2 | — | |
RBWMYPKAPIYTJQ
|
7.8 | IC50 | 2 | — | |
UTSXCJSXSSVXHI
|
7.8 | Ki | 2 | — | |
FHIFVYKWPHPFEV
|
7.8 | IC50 | 4 | — | |
MJZNRHTYZRSATJ
|
7.8 | IC50 | 2 | — | |
AQACCMRPIZQLDS
|
7.8 | Ki | 2 | — | |
SKPHSTUDURJNOT
|
7.8 | Ki | 2 | — | |
FEECZRRIVKANPB
|
7.7 | IC50 | 2 | — | |
NFXZAFCZOMISJH
|
7.7 | IC50 | 2 | — | |
WHELBSIYNGCJSE
|
7.7 | IC50 | 2 | — | |
DVFMRMSQBLLRFB
|
7.7 | IC50 | 3 | — | |
JDNUFWMCDUMKPL
|
7.7 | IC50 | 2 | — | |
QMPBBNUOBOFBFS
|
7.7 | IC50 | 2 | — | |
UNICQUXWGGDNLF
|
7.7 | IC50 | 4 | — | |
UZXUKPUBPQPIQC
|
7.7 | IC50 | 2 | — | |
GRGDWLDSVPJEJU
|
7.7 | IC50 | 2 | — | |
VKELCWVLNDHDSK
|
7.7 | IC50 | 2 | — | |
XQMQPBAYXGGXEY
|
7.7 | IC50 | 2 | — | |
QRTUECBYTYJXHL
|
7.7 | IC50 | 2 | — | |
PTGYXJBPMNPISM
|
7.6 | IC50 | 2 | — | |
WFJHHZOLVBKTCG
|
7.6 | IC50 | 2 | — | |
LTCAMZPTBRHGIT
|
7.6 | IC50 | 4 | — | |
OZCGFUYWRSIHLJ
|
7.6 | IC50 | 2 | — | |
SMQQOJDQJBWRCU
|
7.6 | IC50 | 2 | — | |
WCFBPQPQLAYXFE
|
7.6 | IC50 | 2 | — | |
MNUHXGJUYTWVLU
|
7.6 | IC50 | 2 | — | |
KVMJONNVSMEASA
|
7.6 | IC50 | 4 | — | |
XUHFZJPQDLAZMY
|
7.6 | IC50 | 2 | — | |
GNSONAJPJOULHV
|
7.6 | IC50 | 2 | — | |
KNFARXVTOTYHMG
|
7.6 | IC50 | 4 | — | |
QNRLUURSWJCRAA
|
7.6 | IC50 | 2 | — | |
FBYZCSUBKCAJAK
|
7.5 | IC50 | 2 | — | |
HQHODRFXEHOYNQ
|
7.5 | IC50 | 2 | — | |
PMIGMAKHNBCGBZ
|
7.5 | IC50 | 2 | — | |
YALGKJMDFDSHJZ
|
7.5 | IC50 | 2 | — | |
HNKKKBJAQYQBOC
|
7.4 | IC50 | 2 | — | |
JVSFPWJWCIUVJO
|
7.4 | IC50 | 2 | — | |
MAQWOCWKZDBXGP
|
7.4 | IC50 | 2 | — | |
HWWLPQZHHBGXAB
|
7.4 | IC50 | 2 | — |