Target Details
| UniProt AC | P0DTD1 |
|---|---|
| Gene Symbol | rep |
| Protein Name | Replicase polyprotein 1ab |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13087 (AAA_12) PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF06471 (CoV_ExoN) PF06460 (CoV_Methyltr_2) PF09401 (CoV_NSP10) PF20631 (CoV_NSP13_1B) PF20633 (CoV_NSP13_stalk) PF20632 (CoV_NSP13_ZBD) PF19215 (CoV_NSP15_C) PF19216 (CoV_NSP15_M) PF19219 (CoV_NSP15_N) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF06478 (CoV_RPol_N) PF01661 (Macro) PF05409 (Peptidase_C30) PF00680 (RdRP_1) |
Summary
- Multi-target molecules 387
- Clinical molecules 3
- Avg pChEMBL 6.91
Active Molecules (387)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PKJWLVLOGHATRZ
|
9.0 | IC50 | 3 | — | |
TXFALORVHGHNIZ
|
9.0 | IC50 | 2 | — | |
INWHDRNGZMHXEZ
|
8.7 | IC50 | 2 | — | |
GSUNDMAZJLWTIT
|
8.7 | IC50 | 2 | — | |
JTZZSQYMACOLNN
|
8.6 | IC50 | 6 | — | |
WGNWEPPRWQKSKI
|
8.6 | Ki | 3 | — | |
IBQXXYZTUWXAPY
|
8.6 | IC50 | 2 | — | |
AWSZFCNWIVMPPT
|
8.5 | IC50 | 2 | — | |
LOFFTBAELMOYKZ
|
8.5 | IC50 | 2 | — | |
QZQMFRGAGVCQAU
|
8.5 | Ki | 2 | — | |
QNLMYJJUQPZSSI
|
8.5 | IC50 | 2 | — | |
APTHLSASJXHTAY
|
8.4 | IC50 | 4 | — | |
FBDZPOPZZIODCH
|
8.4 | Ki | 2 | — | |
PXPFKYBINQAOCO
|
8.4 | Ki | 2 | — | |
YFAVHMGYTFULDO
|
8.4 | Ki | 2 | — | |
KQASAMHEMLKUIM
|
8.4 | IC50 | 2 | — | |
CJXNCBSSADROTD
|
8.3 | IC50 | 2 | — | |
MXEGAMGMDDENAC
|
8.3 | Ki | 2 | — | |
WAXJMBFCXYZEEF
|
8.3 | IC50 | 2 | — | |
UIXQHURPUVBNCZ
|
8.3 | IC50 | 2 | — | |
HSSWPCDEWPTIQS
|
8.3 | IC50 | 2 | — | |
QHBWMDVARYUYJW
|
8.3 | IC50 | 2 | — | |
ILOODQHBNBJAAG
|
8.2 | IC50 | 2 | — | |
RRGARHLRSSYTCB
|
8.2 | IC50 | 2 | — | |
ULEIWGQRBVSCTG
|
8.2 | IC50 | 2 | — | |
JWFKMTSCIZNZAE
|
8.2 | IC50 | 2 | — | |
RAAXPKDUFYAXAD
|
8.2 | IC50 | 2 | — | |
PAJZPMREBNPURC
|
8.2 | IC50 | 2 | — | |
RHFOTHRIPKQIDW
|
8.2 | IC50 | 2 | — | |
ULEIWGQRBVSCTG
|
8.2 | IC50 | 2 | — | |
WUMUSTXWZPBYJT
|
8.2 | IC50 | 2 | — | |
DDNKJVYYJPDFOE
|
8.1 | IC50 | 2 | — | |
QFTTVHGJIGPMTG
|
8.1 | IC50 | 2 | — | |
BDSQVYWAMBOWIL
|
8.1 | IC50 | 4 | — | |
VDPJORBKOLOGMZ
|
8.1 | IC50 | 2 | — | |
BFFXBTWXMYGLLP
|
8.1 | IC50 | 2 | — | |
LIENCHBZNNMNKG
|
8.1 | IC50 | 2 | — | |
UGXSZZAITMURED
|
8.1 | IC50 | 2 | — | |
ALCYYDYSILTTKJ
|
8.1 | IC50 | 2 | — | |
DAVWSCGJIBGBHZ
|
8.1 | IC50 | 2 | — | |
JCUWWLFQYPMDMI
|
8.1 | IC50 | 4 | — | |
KRNQXZIZXPQQEL
|
8.1 | Ki | 2 | — | |
PDQAUBWJYWYCIF
|
8.1 | IC50 | 2 | — | |
NCMBMJWVGROMTF
|
8.0 | IC50 | 3 | — | |
GBJVAVGBSGRRKN
|
8.0 | IC50 | 2 | — | |
KSBJTEAOFRKHIW
|
8.0 | IC50 | 2 | — | |
KSSDFKAUXACCMX
|
8.0 | IC50 | 2 | — | |
MMVYUHFDLZLNDJ
|
8.0 | IC50 | 2 | — | |
QMPBBNUOBOFBFS
|
8.0 | IC50 | 2 | — | |
SVOCCYIUNITIHL
|
8.0 | IC50 | 2 | — |