Target Details
| UniProt AC | P0DTC1 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Replicase polyprotein 1a |
| Organism | Severe acute respiratory syndrome coronavirus 2 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF09401 (CoV_NSP10) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF01661 (Macro) PF05409 (Peptidase_C30) |
Summary
- Multi-target molecules 197
- Clinical molecules 0
- Avg pChEMBL 7.1
Active Molecules (197)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GTLDPUSOCDSHIU
|
6.3 | IC50 | 2 | — | |
GZWRFHALZSJWCL
|
6.3 | IC50 | 2 | — | |
HOGIUARUHFASKN
|
6.3 | IC50 | 2 | — | |
HWBPESUHQMIXLB
|
6.3 | IC50 | 2 | — | |
IPGMAZLYVSWCJD
|
6.3 | IC50 | 2 | — | |
JCPOHWPGDQUOQN
|
6.3 | IC50 | 2 | — | |
JLZPYUNNWVRLGQ
|
6.3 | IC50 | 2 | — | |
JLZPYUNNWVRLGQ
|
6.3 | IC50 | 2 | — | |
JSAQCZWEOZMZCG
|
6.3 | IC50 | 2 | — | |
KAPDZTAMKBHBAC
|
6.3 | IC50 | 2 | — | |
KRNGPDUFHQXSOZ
|
6.3 | IC50 | 2 | — | |
LSFMSEYLICBQLD
|
6.3 | IC50 | 2 | — | |
LSFMSEYLICBQLD
|
6.3 | IC50 | 2 | — | |
LUMXDKZMUPIRHM
|
6.3 | IC50 | 2 | — | |
LVLPBPSLLDDHMK
|
6.3 | IC50 | 2 | — | |
MMOGDCKWHZFLMO
|
6.3 | IC50 | 2 | — | |
MRSXETXDOITHNK
|
6.3 | IC50 | 2 | — | |
MVMXSHQQBNAWMC
|
6.3 | IC50 | 2 | — | |
OYEOCKYUCQUKMH
|
6.3 | IC50 | 2 | — | |
OYEOCKYUCQUKMH
|
6.3 | IC50 | 2 | — | |
QFWWLRCXQIIMLA
|
6.3 | IC50 | 2 | — | |
QJDMARSQHXLLBE
|
6.3 | IC50 | 2 | — | |
RCFGNCPIHMGBGF
|
6.3 | IC50 | 2 | — | |
RFISFJYBBQQZPY
|
6.3 | IC50 | 2 | — | |
RUJRCMWJRKOZTO
|
6.3 | IC50 | 2 | — | |
SIQVSLICJZAZGM
|
6.3 | IC50 | 2 | — | |
UEGSTNJPMSGHMF
|
6.3 | IC50 | 2 | — | |
VQJHSXBJTLPKHO
|
6.3 | IC50 | 2 | — | |
VVXBKZFYMWTAHG
|
6.3 | IC50 | 2 | — | |
VYYDFJQUXALHPF
|
6.3 | IC50 | 2 | — | |
VYYDFJQUXALHPF
|
6.3 | IC50 | 2 | — | |
XHWLSZIPRUJMBX
|
6.3 | IC50 | 2 | — | |
XHWLSZIPRUJMBX
|
6.3 | IC50 | 2 | — | |
YCSCOAGMDRJISW
|
6.3 | IC50 | 2 | — | |
ZSSDZVMVWPPHTJ
|
6.3 | IC50 | 2 | — | |
ZZNLHLJRATZLSO
|
6.3 | IC50 | 2 | — | |
QLWOSILDDBBNKU
|
6.2 | Ki | 2 | — | |
ZPEDAVGOVRCNQR
|
6.2 | IC50 | 2 | — | |
FMPUADOXTPMTON
|
6.2 | IC50 | 2 | — | |
MKZYMKKUBVPEET
|
6.2 | Ki | 2 | — | |
RXNNWOBJWBKPHT
|
6.2 | IC50 | 2 | — | |
JZRRCGQQCZGHEA
|
6.1 | IC50 | 2 | — | |
HZTJOSBNLNQPCX
|
6.1 | IC50 | 2 | — | |
WBLZKCOFIDSWKH
|
6.1 | Kd | 2 | — | |
YIEPOGUSSKXXSP
|
6.1 | Ki | 2 | — | |
XCUCLKWBHWYCEZ
|
6.1 | Kd | 2 | — | |
LIENCHBZNNMNKG
|
6.1 | Ki | 2 | — |