Target Details
| UniProt AC | P0C6U8 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Replicase polyprotein 1a |
| Organism | Severe acute respiratory syndrome coronavirus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF12379 (bCoV_NSP3_N) PF12124 (bCoV_SUD_C) PF11633 (bCoV_SUD_M) PF09401 (CoV_NSP10) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF01661 (Macro) PF05409 (Peptidase_C30) |
Summary
- Multi-target molecules 85
- Clinical molecules 0
- Avg pChEMBL 6.62
Active Molecules (85)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FPOUHYIBNRERGL
|
6.2 | IC50 | 2 | — | |
UTDZHTFBLCBKHG
|
6.2 | IC50 | 2 | — | |
UVERBUNNCOKGNZ
|
6.2 | IC50 | 2 | — | |
HEVGAFYDYPEGEP
|
6.2 | Ki | 2 | — | |
NFWQGKLIEDRSFG
|
6.2 | IC50 | 2 | — | |
CMJOQABPDRNNJZ
|
6.2 | Ki | 2 | — | |
KMVKSBHPOAHWOA
|
6.2 | Ki | 2 | — | |
WDMSWWUPIMEGNZ
|
6.2 | Ki | 2 | — | |
YNXKLJCBBNQTSI
|
6.2 | Ki | 2 | — | |
AQIUEOPKDZKYFU
|
6.2 | Ki | 2 | — | |
NDXWDWBHDSNJNP
|
6.2 | IC50 | 2 | — | |
NDXWDWBHDSNJNP
|
6.2 | IC50 | 2 | — | |
NGIZLVDUIAGJQR
|
6.2 | IC50 | 2 | — | |
QDRCGHXOZNVPFX
|
6.2 | Ki | 2 | — | |
UGSXTJOTPOFHOD
|
6.2 | IC50 | 2 | — | |
PDLFIYNGGUUVLF
|
6.1 | Ki | 2 | — | |
QBIWXGCBGBHXON
|
6.1 | IC50 | 2 | — | |
CTJDSJGCDMNHRC
|
6.1 | Kd | 2 | — | |
GEXHQXMZXYXJPR
|
6.1 | Kd | 2 | — | |
QEKGJLUOEDTRIW
|
6.1 | IC50 | 2 | — | |
QIXFKLPOAIIFGF
|
6.1 | IC50 | 2 | — | |
XDKZVJYVKZWDNH
|
6.1 | Ki | 2 | — | |
CFQSYTCHYSNACR
|
6.1 | IC50 | 2 | — | |
SHSPLTGUTOVZEW
|
6.1 | IC50 | 2 | — | |
YGALISXJEIZOHZ
|
6.1 | IC50 | 2 | — | |
QSVAUAVIZAYJHW
|
6.1 | Ki | 2 | — | |
HXYPMMAPDRFFTM
|
6.0 | IC50 | 2 | — | |
NENXLTIJMAMZOM
|
6.0 | IC50 | 2 | — | |
QHXIEOUYOSYVEB
|
6.0 | IC50 | 2 | — | |
WKNCKKOHQQLNCY
|
6.0 | IC50 | 3 | — | |
MAYSJMBSILUGEG
|
6.0 | IC50 | 3 | — | |
IQVFCZXMGASAGI
|
6.0 | IC50 | 2 | — | |
LHBIUOYHJIXRST
|
6.0 | IC50 | 2 | — | |
UFOWXDUBQLPEOX
|
6.0 | IC50 | 2 | — | |
FOLCUFKJHSQMEL
|
6.0 | IC50 | 3 | — |