Target Details
| UniProt AC | P0C1U9 |
|---|---|
| Gene Symbol | parC |
| Protein Name | DNA topoisomerase 4 subunit A |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 57
- Clinical molecules 0
- Avg pChEMBL 6.48
Active Molecules (57)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CEDOVDFAPKPYNH
|
6.1 | IC50 | 4 | — | |
REEOSLJMDKKLQA
|
6.1 | IC50 | 4 | — | |
ZFMCWMJGTDHLKI
|
6.0 | IC50 | 4 | — | |
QOIXLMNVJYVPLA
|
6.0 | IC50 | 4 | — | |
YJGCQIKMBDWQSU
|
6.0 | IC50 | 4 | — | |
JHJANKDCEYKCQY
|
6.0 | IC50 | 4 | — | |
MYSWGUAQZAJSOK
|
6.0 | IC50 | 6 | — |