Target Details
| UniProt AC | P0C1S7 |
|---|---|
| Gene Symbol | parE |
| Protein Name | DNA topoisomerase 4 subunit B |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 52
- Clinical molecules 0
- Avg pChEMBL 6.48
Active Molecules (52)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XMRMYIYEEWALOZ
|
8.1 | IC50 | 4 | — | |
BKUISYCLLXCBJV
|
7.9 | Ki | 4 | — | |
RDTDFCZCBIXFEI
|
7.3 | IC50 | 5 | — | |
COTQDURISRILOR
|
7.2 | IC50 | 2 | — | |
PQWWHNZAZANFOZ
|
7.1 | IC50 | 5 | — | |
IYJZRZIDVYDIHE
|
7.1 | IC50 | 3 | — | |
KLPNELPTKNRMMW
|
7.0 | IC50 | 4 | — | |
TVDNDLRKUKVCCR
|
6.9 | IC50 | 4 | — | |
VINPUJZJRCEBET
|
6.8 | IC50 | 5 | — | |
PHKHNRMHOSCRKO
|
6.7 | IC50 | 4 | — | |
GFQDXSUJWFUHQT
|
6.7 | IC50 | 4 | — | |
ZQRZCLVUOLDFJC
|
6.6 | IC50 | 4 | — | |
ZYUKGEKHLULSGR
|
6.6 | IC50 | 4 | — | |
MCMNYTOHUPZLOA
|
6.6 | IC50 | 5 | — | |
GBQZRFCGAJTKDG
|
6.5 | IC50 | 4 | — | |
RVKKBUSSKLNKTC
|
6.5 | IC50 | 4 | — | |
IDBNSMFFTLKKMN
|
6.5 | IC50 | 4 | — | |
USGHRRVFKSLEJT
|
6.5 | IC50 | 4 | — | |
ASSSIFUQVIZHMH
|
6.5 | IC50 | 4 | — | |
VSRUEFVCYYXLCL
|
6.5 | IC50 | 4 | — | |
NHXTWWVJRWMAAW
|
6.5 | IC50 | 4 | — | |
CLAOMDJUURAQOM
|
6.5 | IC50 | 4 | — | |
YERDVHADHPXHFF
|
6.4 | IC50 | 4 | — | |
CDWUOIQIYZWIIH
|
6.4 | IC50 | 2 | — | |
HVMVZISHQKEBLK
|
6.4 | IC50 | 4 | — | |
PNXMNHGKWCLCMU
|
6.4 | IC50 | 4 | — | |
NCIFTFPQZBACJB
|
6.4 | IC50 | 2 | — | |
GUEBWQFTJDQZMH
|
6.3 | IC50 | 2 | — | |
NTNKQRBKOGURQE
|
6.3 | IC50 | 4 | — | |
PEKRPORMYGTOHQ
|
6.3 | IC50 | 4 | — | |
TWOGVSMCVZUIJI
|
6.3 | IC50 | 4 | — | |
XTVIZXPGQNSAAD
|
6.3 | IC50 | 4 | — | |
ZIEKVRDXDUZMKV
|
6.3 | IC50 | 4 | — | |
NIIWFDOFEHUZBO
|
6.3 | IC50 | 4 | — | |
MYSWGUAQZAJSOK
|
6.3 | IC50 | 6 | — | |
SHKVDXCLBNOXFB
|
6.2 | IC50 | 4 | — | |
DLXOHRWBSQWBAJ
|
6.2 | IC50 | 2 | — | |
JRAGTUWUNIDVFX
|
6.2 | IC50 | 4 | — | |
KDGQBAIMBSYHIS
|
6.2 | IC50 | 4 | — | |
PZFAZQUREQIODZ
|
6.2 | IC50 | 4 | — | |
QMBIGGCLOHYBHN
|
6.2 | IC50 | 4 | — | |
RXPOVSSVBGRCOL
|
6.2 | IC50 | 4 | — | |
YJGCQIKMBDWQSU
|
6.2 | IC50 | 4 | — | |
IJZXBWJKPBRXAR
|
6.1 | IC50 | 4 | — | |
QUDWUIDMIRCCRB
|
6.1 | IC50 | 4 | — | |
NHLOTGIWHZMOCX
|
6.1 | IC50 | 3 | — | |
CEDOVDFAPKPYNH
|
6.1 | IC50 | 4 | — | |
REEOSLJMDKKLQA
|
6.1 | IC50 | 4 | — | |
ZFMCWMJGTDHLKI
|
6.0 | IC50 | 4 | — | |
QOIXLMNVJYVPLA
|
6.0 | IC50 | 4 | — |