Target Details
| UniProt AC | P0AES6 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF21249 (GyrB_hook) PF18053 (GyrB_insert) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 337
- Clinical molecules 0
- Avg pChEMBL 7.06
Active Molecules (337)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HXYBRUDRPDMKEK
|
6.1 | IC50 | 2 | — | |
KZVFTFMKZAUXKO
|
6.1 | IC50 | 2 | — | |
MOFJXSJDPANQFX
|
6.1 | IC50 | 2 | — | |
PXANBKOATAYLNW
|
6.1 | IC50 | 2 | — | |
SOKJBFLDJIUGCW
|
6.1 | IC50 | 2 | — | |
SVKKHTJYMQDGDV
|
6.1 | IC50 | 2 | — | |
VSPOWGLFXRJICV
|
6.1 | IC50 | 2 | — | |
YMYSBGNTLMKPJD
|
6.1 | IC50 | 2 | — | |
PDRCNKSNILMXSD
|
6.1 | IC50 | 2 | — | |
KXDJSAAYOSJRNC
|
6.1 | IC50 | 2 | — | |
DFIJENIBCXNIGZ
|
6.0 | IC50 | 2 | — | |
DRHQZOCCHAGCFJ
|
6.0 | IC50 | 2 | — | |
FRSGMLIUXXMDRV
|
6.0 | IC50 | 2 | — | |
HOZCTRWTVFKGBZ
|
6.0 | IC50 | 2 | — | |
HUQYMKUZMWKXSJ
|
6.0 | IC50 | 2 | — | |
PGEIHRYPSMAENW
|
6.0 | IC50 | 2 | — | |
PVNOUCKOXQSARZ
|
6.0 | IC50 | 2 | — | |
RELYTUGZZNYKPH
|
6.0 | IC50 | 2 | — | |
USIMQOIUWHIQOV
|
6.0 | IC50 | 2 | — | |
YCVBALOHZCSOAU
|
6.0 | IC50 | 2 | — | |
FTJURNSPWPKGJD
|
6.0 | IC50 | 2 | — | |
NCTPTGLNCLEXKF
|
6.0 | IC50 | 2 | — | |
YIVGSUPJSMHNEV
|
6.0 | IC50 | 2 | — | |
PNZRVUNLSZGZSV
|
6.0 | IC50 | 2 | — | |
FIFPIKDNMUSOAF
|
6.0 | IC50 | 2 | — | |
JTGPFBMJIYJYNZ
|
6.0 | IC50 | 2 | — | |
MKHBXCHRTDKRFA
|
6.0 | IC50 | 2 | — | |
OCFPRHXENHKVOI
|
6.0 | IC50 | 2 | — | |
RYGQUNHPYQJBTQ
|
6.0 | IC50 | 2 | — | |
STERFRCBIKXRFO
|
6.0 | IC50 | 2 | — | |
SWDVPSPYHLMYHA
|
6.0 | IC50 | 2 | — | |
VJWYBRYEYKPJOT
|
6.0 | IC50 | 2 | — | |
VOYUBWQGNLEVQI
|
6.0 | IC50 | 2 | — | |
VSKMXQVCZULPKO
|
6.0 | IC50 | 2 | — | |
XMILWIODYWNKFR
|
6.0 | IC50 | 2 | — | |
YWJJMGOABBHKMZ
|
6.0 | IC50 | 2 | — | |
ZUBLOLWIOGHOAF
|
6.0 | IC50 | 2 | — |