Target Details
| UniProt AC | P0AES6 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF21249 (GyrB_hook) PF18053 (GyrB_insert) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 337
- Clinical molecules 0
- Avg pChEMBL 7.06
Active Molecules (337)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ATBBCOJFLILWTN
|
6.3 | IC50 | 2 | — | |
JDRIHSSGXXPQER
|
6.3 | IC50 | 2 | — | |
LOCOAFTWPSEOFN
|
6.3 | IC50 | 2 | — | |
LXWWGDMZJZNTAM
|
6.3 | IC50 | 2 | — | |
MBCCAHOCJOACSK
|
6.3 | IC50 | 2 | — | |
ONQJCPZRYFXJAT
|
6.3 | IC50 | 2 | — | |
RCBUOEVVPLRUIV
|
6.3 | IC50 | 2 | — | |
SKFJUUFDRKDKRK
|
6.3 | IC50 | 2 | — | |
SVQBHXGGUYGYIA
|
6.3 | IC50 | 2 | — | |
VGOVVJRVKIMXAH
|
6.3 | IC50 | 2 | — | |
XAJJUFKXNKKIQI
|
6.3 | IC50 | 2 | — | |
XUBOMFCQGDBHNK
|
6.3 | IC50 | 2 | — | |
YYWLDHVFBDQOSB
|
6.3 | IC50 | 2 | — | |
ZRCVYEYHRGVLOC
|
6.3 | IC50 | 3 | — | |
CLAOMDJUURAQOM
|
6.3 | IC50 | 4 | — | |
MZMZOPRUDJUCTH
|
6.3 | IC50 | 2 | — | |
YQYCIWQOVOMHTE
|
6.3 | IC50 | 2 | — | |
PKZNGTXURVSDRW
|
6.2 | IC50 | 2 | — | |
XJAPVFDVPQVNTP
|
6.2 | IC50 | 2 | — | |
QALHKQTVOWHLQA
|
6.2 | IC50 | 2 | — | |
BIWANTQRBZHDNP
|
6.2 | IC50 | 2 | — | |
DAIBUTBYIXSWIF
|
6.2 | IC50 | 2 | — | |
IQFVZJHGVZQCBU
|
6.2 | IC50 | 2 | — | |
JYTKLNNKDJTVJR
|
6.2 | IC50 | 2 | — | |
MMBOMVDEWMUTNS
|
6.2 | IC50 | 2 | — | |
MZJHEYLDFYCQTG
|
6.2 | IC50 | 2 | — | |
NXCNASGAEQGJFI
|
6.2 | IC50 | 2 | — | |
OGJPXUAPXNRGGI
|
6.2 | IC50 | 3 | — | |
QBEKDHJCXXJSMG
|
6.2 | IC50 | 2 | — | |
QRLSRELXQXBCKO
|
6.2 | IC50 | 2 | — | |
XYUDRALUFQLYQD
|
6.2 | IC50 | 2 | — | |
NPFVTDFFMCQGEY
|
6.2 | IC50 | 2 | — | |
OLZJUUMILDSQRJ
|
6.2 | IC50 | 2 | — | |
CORWQFLKJCXVKC
|
6.2 | IC50 | 2 | — | |
RGSYWFKWPTYADN
|
6.2 | IC50 | 2 | — | |
DTLIOBULPHFNCN
|
6.2 | IC50 | 2 | — | |
BYTLKESUZQQJMP
|
6.2 | IC50 | 2 | — | |
IBCYSYSDUXVMHM
|
6.2 | IC50 | 2 | — | |
KFRZFWRNTZMYGG
|
6.2 | IC50 | 2 | — | |
LIGLNYMZXUCCIB
|
6.2 | IC50 | 2 | — | |
LLXAFYKXFAACNG
|
6.2 | IC50 | 2 | — | |
PKSRQRFDRMZEJO
|
6.2 | IC50 | 2 | — | |
SMUYQNDYNHLRPO
|
6.2 | IC50 | 2 | — | |
VIIQSEKXRPSHBZ
|
6.2 | IC50 | 2 | — | |
YXMRPTNKUBGVMH
|
6.2 | IC50 | 2 | — | |
ZDYYFHJCQVAOBA
|
6.2 | IC50 | 2 | — | |
UOFAYEAZDTZGPQ
|
6.1 | IC50 | 2 | — | |
BGTMVPCTKSRAIT
|
6.1 | IC50 | 2 | — | |
DBHRNNUAKNLSTN
|
6.1 | IC50 | 2 | — | |
FXNYDQUBEWWQKM
|
6.1 | IC50 | 2 | — |