Target Details
| UniProt AC | P0AES6 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF21249 (GyrB_hook) PF18053 (GyrB_insert) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 337
- Clinical molecules 0
- Avg pChEMBL 7.06
Active Molecules (337)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVJWLIUONXIZCV
|
6.7 | IC50 | 2 | — | |
XRTAULGTMMIAID
|
6.7 | IC50 | 2 | — | |
XLGIJKUFLIGITI
|
6.7 | IC50 | 2 | — | |
QNIRZGVLRPNLDU
|
6.7 | IC50 | 2 | — | |
CPTVFJTVHOYDTL
|
6.6 | IC50 | 2 | — | |
QULNBEHUNMRDOZ
|
6.6 | IC50 | 2 | — | |
OFYFNDCPZYDSHV
|
6.6 | IC50 | 2 | — | |
JJXHHUOQDCCPHY
|
6.6 | IC50 | 2 | — | |
DSRDRGMPVRBOFT
|
6.5 | IC50 | 2 | — | |
SWKYJQWWRWIUFS
|
6.5 | IC50 | 2 | — | |
ULHHEGLIKLUVMD
|
6.5 | IC50 | 2 | — | |
HJXNKCZQPUWIPK
|
6.5 | IC50 | 2 | — | |
LQUTWAXMKCCOBE
|
6.5 | IC50 | 2 | — | |
CAVIKQQEXPNJNV
|
6.5 | IC50 | 2 | — | |
FABPRXSRWADJSP
|
6.5 | IC50 | 3 | — | |
FWKBFPFKHVTISW
|
6.5 | IC50 | 2 | — | |
GQTOYQNDZQOUHI
|
6.5 | IC50 | 2 | — | |
HFRGSVIKEOBJHY
|
6.5 | IC50 | 2 | — | |
JYDZVUWVVASPRQ
|
6.5 | IC50 | 2 | — | |
KHXIOPHRPYYECT
|
6.5 | IC50 | 2 | — | |
MYSWGUAQZAJSOK
|
6.5 | IC50 | 6 | — | |
OQSLKWQIYRYOKJ
|
6.5 | IC50 | 2 | — | |
POTUKOMZFDWDHQ
|
6.5 | IC50 | 2 | — | |
QKEHSEZUBTWJJC
|
6.5 | IC50 | 2 | — | |
RYOHJGVWLGKRGX
|
6.5 | IC50 | 2 | — | |
TZQOEAUYWDIUHZ
|
6.5 | IC50 | 2 | — | |
VIVDPWOYADDJAN
|
6.5 | IC50 | 2 | — | |
XOAFVAOSKYSOIS
|
6.5 | IC50 | 2 | — | |
QKEHSEZUBTWJJC
|
6.5 | IC50 | 2 | — | |
SEEBUHTYKMBMPL
|
6.5 | IC50 | 2 | — | |
ZTIMRGPSOAADPP
|
6.5 | IC50 | 2 | — | |
ZJOVVADZPGXOGF
|
6.5 | IC50 | 2 | — | |
SBWCMUMKNBMKNA
|
6.4 | IC50 | 2 | — | |
YUFDLDKPRBELKV
|
6.4 | IC50 | 2 | — | |
JDBFQWHOEJRPES
|
6.4 | IC50 | 2 | — | |
KSKYADHIJGMLQL
|
6.4 | IC50 | 2 | — | |
NLPBUFDDDFGFJO
|
6.4 | IC50 | 2 | — | |
SQDSWGQSOYDJPW
|
6.4 | IC50 | 2 | — | |
XDNYDODHLMBYAK
|
6.4 | IC50 | 2 | — | |
YUFDLDKPRBELKV
|
6.4 | IC50 | 2 | — | |
ZJSPGPLJDRIYLI
|
6.4 | IC50 | 2 | — | |
GAHLNYQPFMZGDZ
|
6.4 | IC50 | 2 | — | |
MGVRFBQCOIBSHZ
|
6.4 | IC50 | 2 | — | |
YZTJFBSSKZKNMR
|
6.4 | IC50 | 2 | — | |
JKSZENONXRNKSS
|
6.4 | IC50 | 2 | — | |
JONHESQYKRXXHZ
|
6.4 | IC50 | 2 | — | |
ZQRZCLVUOLDFJC
|
6.4 | IC50 | 4 | — | |
PVCLTSIILIOCFZ
|
6.3 | IC50 | 2 | — | |
OHJASJJMGQDYNR
|
6.3 | IC50 | 2 | — | |
AQJPWQPUBWBDQE
|
6.3 | IC50 | 2 | — |