Target Details
| UniProt AC | P0AES6 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF21249 (GyrB_hook) PF18053 (GyrB_insert) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 337
- Clinical molecules 0
- Avg pChEMBL 7.06
Active Molecules (337)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KOVLKWGJIYFSRO
|
8.1 | IC50 | 2 | — | |
RSCJTJIKINXWDW
|
8.1 | IC50 | 2 | — | |
MBCOBCDFYMQNQZ
|
8.1 | IC50 | 2 | — | |
SZIOCYHUCPYPPG
|
8.1 | IC50 | 2 | — | |
DBXSXNHVESUPOA
|
8.0 | IC50 | 2 | — | |
AAWYAFMPUFDEST
|
8.0 | IC50 | 2 | — | |
YJGCQIKMBDWQSU
|
8.0 | IC50 | 4 | — | |
TWQUSFPXFBUZAU
|
8.0 | IC50 | 2 | — | |
UMVFQZONUAUFGC
|
8.0 | IC50 | 2 | — | |
KAIGENGZIZRWMW
|
7.9 | IC50 | 2 | — | |
FWKBFPFKHVTISW
|
7.9 | IC50 | 2 | — | |
JXMRFLWUZASPFL
|
7.9 | IC50 | 2 | — | |
ZKNZKHAAVPVEAJ
|
7.9 | IC50 | 2 | — | |
GILVJABPOPBFRB
|
7.8 | IC50 | 2 | — | |
JETKTBLDFMGAOL
|
7.8 | IC50 | 2 | — | |
NKCCKBBSHMGYMD
|
7.8 | IC50 | 2 | — | |
IIGBANOVZFEHJC
|
7.8 | IC50 | 2 | — | |
XZLCLAKXNCMYKU
|
7.8 | IC50 | 2 | — | |
BYYFORUHJRHMMU
|
7.8 | IC50 | 2 | — | |
BYYFORUHJRHMMU
|
7.8 | IC50 | 2 | — | |
IEHUSEXPEOJDEF
|
7.8 | IC50 | 2 | — | |
YFRGLVPTZHJWIM
|
7.8 | IC50 | 2 | — | |
RLIDZVBFXZCVEH
|
7.8 | IC50 | 2 | — | |
FSOAZMGZMXDGQX
|
7.7 | IC50 | 2 | — | |
VLCKPYIQPLGTCI
|
7.7 | IC50 | 2 | — | |
OYTVSJBMPLZYQI
|
7.7 | IC50 | 2 | — | |
VQYUKJQPDIGREC
|
7.7 | IC50 | 2 | — | |
YOFXMMYBDPSZAB
|
7.7 | IC50 | 2 | — | |
LGQLJKHATNDFOW
|
7.7 | IC50 | 2 | — | |
RXANXGVEULKMLY
|
7.7 | IC50 | 3 | — | |
BGZNIXFHOSDNBY
|
7.7 | IC50 | 2 | — | |
AMYYSRVSJKCUAD
|
7.6 | IC50 | 2 | — | |
HKGIQYKOHZBOTG
|
7.6 | IC50 | 2 | — | |
FWKBFPFKHVTISW
|
7.6 | IC50 | 2 | — | |
HIZAXRZCORUSNT
|
7.6 | IC50 | 2 | — | |
OTIMTRNHWWKMHS
|
7.6 | IC50 | 2 | — | |
REMFYECIOFGXBB
|
7.6 | IC50 | 2 | — | |
GAUTWGMJXMALGW
|
7.5 | IC50 | 2 | — | |
QOIXLMNVJYVPLA
|
7.5 | IC50 | 4 | — | |
WNWGHNNOTRTXOM
|
7.5 | IC50 | 2 | — | |
QISBQJCTBKCLRU
|
7.5 | IC50 | 2 | — | |
KYOIGEZIXURVNO
|
7.5 | IC50 | 2 | — | |
OZDLVAWIASMACL
|
7.5 | IC50 | 2 | — | |
UNPWBBYTMMYTPY
|
7.4 | IC50 | 3 | — | |
MHDUFODFABPRAE
|
7.4 | IC50 | 2 | — | |
FAKRMULLXOZHQH
|
7.4 | IC50 | 2 | — | |
IPGUFGCGLXUDOJ
|
7.4 | IC50 | 2 | — | |
RVKZOHUACTYRCJ
|
7.4 | IC50 | 2 | — | |
GEDDMFGBKRREEU
|
7.4 | IC50 | 2 | — | |
XKRJEBDYVJJENF
|
7.4 | IC50 | 2 | — |