Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LIGLNYMZXUCCIB
|
6.2 | IC50 | 2 | — | |
LLXAFYKXFAACNG
|
6.2 | IC50 | 2 | — | |
PKSRQRFDRMZEJO
|
6.2 | IC50 | 2 | — | |
SMUYQNDYNHLRPO
|
6.2 | IC50 | 2 | — | |
VIIQSEKXRPSHBZ
|
6.2 | IC50 | 2 | — | |
YXMRPTNKUBGVMH
|
6.2 | IC50 | 2 | — | |
ZDYYFHJCQVAOBA
|
6.2 | IC50 | 2 | — | |
UOFAYEAZDTZGPQ
|
6.1 | IC50 | 2 | — | |
BGTMVPCTKSRAIT
|
6.1 | IC50 | 2 | — | |
DBHRNNUAKNLSTN
|
6.1 | IC50 | 2 | — | |
FXNYDQUBEWWQKM
|
6.1 | IC50 | 2 | — | |
HXYBRUDRPDMKEK
|
6.1 | IC50 | 2 | — | |
KZVFTFMKZAUXKO
|
6.1 | IC50 | 2 | — | |
MOFJXSJDPANQFX
|
6.1 | IC50 | 2 | — | |
PXANBKOATAYLNW
|
6.1 | IC50 | 2 | — | |
SOKJBFLDJIUGCW
|
6.1 | IC50 | 2 | — | |
SVKKHTJYMQDGDV
|
6.1 | IC50 | 2 | — | |
VSPOWGLFXRJICV
|
6.1 | IC50 | 2 | — | |
YMYSBGNTLMKPJD
|
6.1 | IC50 | 2 | — | |
PDRCNKSNILMXSD
|
6.1 | IC50 | 2 | — | |
KXDJSAAYOSJRNC
|
6.1 | IC50 | 2 | — | |
DFIJENIBCXNIGZ
|
6.0 | IC50 | 2 | — | |
DRHQZOCCHAGCFJ
|
6.0 | IC50 | 2 | — | |
FRSGMLIUXXMDRV
|
6.0 | IC50 | 2 | — | |
HOZCTRWTVFKGBZ
|
6.0 | IC50 | 2 | — | |
HUQYMKUZMWKXSJ
|
6.0 | IC50 | 2 | — | |
PGEIHRYPSMAENW
|
6.0 | IC50 | 2 | — | |
PVNOUCKOXQSARZ
|
6.0 | IC50 | 2 | — | |
RELYTUGZZNYKPH
|
6.0 | IC50 | 2 | — | |
USIMQOIUWHIQOV
|
6.0 | IC50 | 2 | — | |
YCVBALOHZCSOAU
|
6.0 | IC50 | 2 | — | |
FTJURNSPWPKGJD
|
6.0 | IC50 | 2 | — | |
NCTPTGLNCLEXKF
|
6.0 | IC50 | 2 | — | |
YIVGSUPJSMHNEV
|
6.0 | IC50 | 2 | — | |
PNZRVUNLSZGZSV
|
6.0 | IC50 | 2 | — | |
FIFPIKDNMUSOAF
|
6.0 | IC50 | 2 | — | |
JTGPFBMJIYJYNZ
|
6.0 | IC50 | 2 | — | |
MKHBXCHRTDKRFA
|
6.0 | IC50 | 2 | — | |
OCFPRHXENHKVOI
|
6.0 | IC50 | 2 | — | |
RYGQUNHPYQJBTQ
|
6.0 | IC50 | 2 | — | |
STERFRCBIKXRFO
|
6.0 | IC50 | 2 | — | |
SWDVPSPYHLMYHA
|
6.0 | IC50 | 2 | — | |
VJWYBRYEYKPJOT
|
6.0 | IC50 | 2 | — | |
VOYUBWQGNLEVQI
|
6.0 | IC50 | 2 | — | |
VSKMXQVCZULPKO
|
6.0 | IC50 | 2 | — | |
XMILWIODYWNKFR
|
6.0 | IC50 | 2 | — | |
YWJJMGOABBHKMZ
|
6.0 | IC50 | 2 | — | |
ZUBLOLWIOGHOAF
|
6.0 | IC50 | 2 | — |