Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUFDLDKPRBELKV
|
6.4 | IC50 | 2 | — | |
ZJSPGPLJDRIYLI
|
6.4 | IC50 | 2 | — | |
GAHLNYQPFMZGDZ
|
6.4 | IC50 | 2 | — | |
MGVRFBQCOIBSHZ
|
6.4 | IC50 | 2 | — | |
YZTJFBSSKZKNMR
|
6.4 | IC50 | 2 | — | |
JKSZENONXRNKSS
|
6.4 | IC50 | 2 | — | |
JONHESQYKRXXHZ
|
6.4 | IC50 | 2 | — | |
ZQRZCLVUOLDFJC
|
6.4 | IC50 | 4 | — | |
PVCLTSIILIOCFZ
|
6.3 | IC50 | 2 | — | |
OHJASJJMGQDYNR
|
6.3 | IC50 | 2 | — | |
AQJPWQPUBWBDQE
|
6.3 | IC50 | 2 | — | |
ATBBCOJFLILWTN
|
6.3 | IC50 | 2 | — | |
JDRIHSSGXXPQER
|
6.3 | IC50 | 2 | — | |
LOCOAFTWPSEOFN
|
6.3 | IC50 | 2 | — | |
LXWWGDMZJZNTAM
|
6.3 | IC50 | 2 | — | |
MBCCAHOCJOACSK
|
6.3 | IC50 | 2 | — | |
ONQJCPZRYFXJAT
|
6.3 | IC50 | 2 | — | |
RCBUOEVVPLRUIV
|
6.3 | IC50 | 2 | — | |
SKFJUUFDRKDKRK
|
6.3 | IC50 | 2 | — | |
SVQBHXGGUYGYIA
|
6.3 | IC50 | 2 | — | |
VGOVVJRVKIMXAH
|
6.3 | IC50 | 2 | — | |
XAJJUFKXNKKIQI
|
6.3 | IC50 | 2 | — | |
XUBOMFCQGDBHNK
|
6.3 | IC50 | 2 | — | |
YYWLDHVFBDQOSB
|
6.3 | IC50 | 2 | — | |
ZRCVYEYHRGVLOC
|
6.3 | IC50 | 3 | — | |
CLAOMDJUURAQOM
|
6.3 | IC50 | 4 | — | |
MZMZOPRUDJUCTH
|
6.3 | IC50 | 2 | — | |
YQYCIWQOVOMHTE
|
6.3 | IC50 | 2 | — | |
PKZNGTXURVSDRW
|
6.2 | IC50 | 2 | — | |
XJAPVFDVPQVNTP
|
6.2 | IC50 | 2 | — | |
QALHKQTVOWHLQA
|
6.2 | IC50 | 2 | — | |
BIWANTQRBZHDNP
|
6.2 | IC50 | 2 | — | |
DAIBUTBYIXSWIF
|
6.2 | IC50 | 2 | — | |
IQFVZJHGVZQCBU
|
6.2 | IC50 | 2 | — | |
JYTKLNNKDJTVJR
|
6.2 | IC50 | 2 | — | |
MMBOMVDEWMUTNS
|
6.2 | IC50 | 2 | — | |
MZJHEYLDFYCQTG
|
6.2 | IC50 | 2 | — | |
NXCNASGAEQGJFI
|
6.2 | IC50 | 2 | — | |
OGJPXUAPXNRGGI
|
6.2 | IC50 | 3 | — | |
QBEKDHJCXXJSMG
|
6.2 | IC50 | 2 | — | |
QRLSRELXQXBCKO
|
6.2 | IC50 | 2 | — | |
XYUDRALUFQLYQD
|
6.2 | IC50 | 2 | — | |
NPFVTDFFMCQGEY
|
6.2 | IC50 | 2 | — | |
OLZJUUMILDSQRJ
|
6.2 | IC50 | 2 | — | |
CORWQFLKJCXVKC
|
6.2 | IC50 | 2 | — | |
RGSYWFKWPTYADN
|
6.2 | IC50 | 2 | — | |
DTLIOBULPHFNCN
|
6.2 | IC50 | 2 | — | |
BYTLKESUZQQJMP
|
6.2 | IC50 | 2 | — | |
IBCYSYSDUXVMHM
|
6.2 | IC50 | 2 | — | |
KFRZFWRNTZMYGG
|
6.2 | IC50 | 2 | — |