Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BNAWAMPTLLVBEW
|
6.7 | IC50 | 2 | — | |
DTSZSZVCLBBHLN
|
6.7 | IC50 | 2 | — | |
FFAHILXYKGISJH
|
6.7 | IC50 | 2 | — | |
JDCMLARRFAPCSR
|
6.7 | IC50 | 2 | — | |
KJYUREWZIBXAOV
|
6.7 | IC50 | 2 | — | |
LUKHUCAYOINUOH
|
6.7 | IC50 | 2 | — | |
LXWREGNACMAAMY
|
6.7 | IC50 | 2 | — | |
RFAPGAPICNQXOM
|
6.7 | IC50 | 2 | — | |
SMONLCFJGCJROJ
|
6.7 | IC50 | 2 | — | |
UVJWLIUONXIZCV
|
6.7 | IC50 | 2 | — | |
XRTAULGTMMIAID
|
6.7 | IC50 | 2 | — | |
XLGIJKUFLIGITI
|
6.7 | IC50 | 2 | — | |
QNIRZGVLRPNLDU
|
6.7 | IC50 | 2 | — | |
CPTVFJTVHOYDTL
|
6.6 | IC50 | 2 | — | |
QULNBEHUNMRDOZ
|
6.6 | IC50 | 2 | — | |
OFYFNDCPZYDSHV
|
6.6 | IC50 | 2 | — | |
JJXHHUOQDCCPHY
|
6.6 | IC50 | 2 | — | |
DSRDRGMPVRBOFT
|
6.5 | IC50 | 2 | — | |
SWKYJQWWRWIUFS
|
6.5 | IC50 | 2 | — | |
ULHHEGLIKLUVMD
|
6.5 | IC50 | 2 | — | |
HJXNKCZQPUWIPK
|
6.5 | IC50 | 2 | — | |
LQUTWAXMKCCOBE
|
6.5 | IC50 | 2 | — | |
CAVIKQQEXPNJNV
|
6.5 | IC50 | 2 | — | |
FABPRXSRWADJSP
|
6.5 | IC50 | 3 | — | |
FWKBFPFKHVTISW
|
6.5 | IC50 | 2 | — | |
GQTOYQNDZQOUHI
|
6.5 | IC50 | 2 | — | |
HFRGSVIKEOBJHY
|
6.5 | IC50 | 2 | — | |
JYDZVUWVVASPRQ
|
6.5 | IC50 | 2 | — | |
KHXIOPHRPYYECT
|
6.5 | IC50 | 2 | — | |
OQSLKWQIYRYOKJ
|
6.5 | IC50 | 2 | — | |
POTUKOMZFDWDHQ
|
6.5 | IC50 | 2 | — | |
QKEHSEZUBTWJJC
|
6.5 | IC50 | 2 | — | |
RGCXUJSMRUJKKB
|
6.5 | IC50 | 2 | — | |
RYOHJGVWLGKRGX
|
6.5 | IC50 | 2 | — | |
TZQOEAUYWDIUHZ
|
6.5 | IC50 | 2 | — | |
XOAFVAOSKYSOIS
|
6.5 | IC50 | 2 | — | |
HLSAPWPGQUYJIF
|
6.5 | IC50 | 2 | — | |
VIVDPWOYADDJAN
|
6.5 | IC50 | 2 | — | |
QKEHSEZUBTWJJC
|
6.5 | IC50 | 2 | — | |
SEEBUHTYKMBMPL
|
6.5 | IC50 | 2 | — | |
ZTIMRGPSOAADPP
|
6.5 | IC50 | 2 | — | |
ZJOVVADZPGXOGF
|
6.5 | IC50 | 2 | — | |
SBWCMUMKNBMKNA
|
6.4 | IC50 | 2 | — | |
YUFDLDKPRBELKV
|
6.4 | IC50 | 2 | — | |
JDBFQWHOEJRPES
|
6.4 | IC50 | 2 | — | |
KSKYADHIJGMLQL
|
6.4 | IC50 | 2 | — | |
NLPBUFDDDFGFJO
|
6.4 | IC50 | 2 | — | |
NPQDLAMGUSTRMY
|
6.4 | Ki | 3 | — | |
SQDSWGQSOYDJPW
|
6.4 | IC50 | 2 | — | |
XDNYDODHLMBYAK
|
6.4 | IC50 | 2 | — |