Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FXVJVTDGWQCYOQ
|
7.0 | IC50 | 3 | — | |
JRMYGOQEFDLQJN
|
7.0 | IC50 | 2 | — | |
KCZWEDWQXOSEMZ
|
7.0 | IC50 | 2 | — | |
KGFYQRFZYURLEH
|
7.0 | IC50 | 2 | — | |
OVFAKDMDTKPFEZ
|
7.0 | IC50 | 2 | — | |
QUQVJLZKLBCCJP
|
7.0 | IC50 | 2 | — | |
UKPJMVBWJKUYSS
|
7.0 | IC50 | 2 | — | |
XQEFOQFUHGWPSD
|
7.0 | IC50 | 2 | — | |
NWDCVIJLQIDCBY
|
7.0 | IC50 | 2 | — | |
LJDGUSFBONSVGJ
|
7.0 | IC50 | 2 | — | |
RVKKBUSSKLNKTC
|
7.0 | IC50 | 4 | — | |
ULKAYELTWNLYQI
|
7.0 | IC50 | 2 | — | |
ZQPFFMNJTDZTRE
|
7.0 | IC50 | 2 | — | |
QEXLBJRFQBGWAC
|
6.9 | IC50 | 2 | — | |
AARJHMDWLTVIEN
|
6.9 | IC50 | 2 | — | |
HLSAPWPGQUYJIF
|
6.9 | IC50 | 2 | — | |
LEZKBUPOVDJOKP
|
6.9 | IC50 | 2 | — | |
OWSXADXRECOTSE
|
6.9 | IC50 | 2 | — | |
PZFAZQUREQIODZ
|
6.9 | IC50 | 4 | — | |
RGGQDRQYPLQVTQ
|
6.9 | IC50 | 2 | — | |
VBIBYFOASQLXQR
|
6.9 | IC50 | 2 | — | |
WCAKRNHRTODWJW
|
6.9 | IC50 | 2 | — | |
XFTTVFZHMRAGMV
|
6.9 | IC50 | 2 | — | |
SIJUCHAWQHDVQI
|
6.9 | Ki | 2 | — | |
WTBABPYUOQESGW
|
6.9 | IC50 | 2 | — | |
ITZFUHUBHMJITR
|
6.9 | IC50 | 2 | — | |
MHWAJESHXFEOOW
|
6.8 | IC50 | 2 | — | |
NEUBWAWYTMZOPY
|
6.8 | IC50 | 2 | — | |
RCYDVAAQJRSRLL
|
6.8 | IC50 | 2 | — | |
UXRKAFKRTDVSDX
|
6.8 | IC50 | 2 | — | |
LYIMJKFUHYOWBM
|
6.8 | IC50 | 2 | — | |
NULLOLQKFUOFDL
|
6.8 | IC50 | 2 | — | |
NWKITMVHAGNKIP
|
6.8 | IC50 | 2 | — | |
RESOFBUAPMFEDQ
|
6.8 | IC50 | 2 | — | |
XTOBVHZEYFCCQZ
|
6.8 | IC50 | 2 | — | |
GXNUHOMLWCVICO
|
6.8 | IC50 | 2 | — | |
HCXCXUYRFPJWRR
|
6.8 | IC50 | 2 | — | |
HHSLFPVGKCXEOG
|
6.8 | IC50 | 2 | — | |
MNRUGEWQKLTAPC
|
6.8 | IC50 | 2 | — | |
UKWCXXCCJYUTTM
|
6.8 | IC50 | 2 | — | |
BYJVKFSAPUBGBY
|
6.8 | IC50 | 2 | — | |
HLSAPWPGQUYJIF
|
6.8 | IC50 | 2 | — | |
PAQUBBVFIYHPDN
|
6.8 | IC50 | 2 | — | |
QUAGKXQUSMJFAP
|
6.8 | IC50 | 2 | — | |
AGUZQNDLLPHGDQ
|
6.8 | IC50 | 2 | — | |
JZFBPMAIHOMKKF
|
6.8 | IC50 | 2 | — | |
TUXCPGXDTVELQJ
|
6.8 | IC50 | 2 | — | |
CASYEBIPRAWOTH
|
6.7 | IC50 | 2 | — | |
TYUGIMHBLIPLKX
|
6.7 | IC50 | 2 | — | |
AEUCESUJMHGFMP
|
6.7 | IC50 | 2 | — |