Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ATNSPUQRDBKCOK
|
7.4 | IC50 | 2 | — | |
HVRAENIVOUQQRG
|
7.4 | IC50 | 2 | — | |
JYRPVRZEIIVAOS
|
7.3 | IC50 | 2 | — | |
NHLOTGIWHZMOCX
|
7.3 | IC50 | 3 | — | |
POYAREGLPUZENY
|
7.3 | IC50 | 2 | — | |
DOXZBGAFRVXDBN
|
7.3 | IC50 | 2 | — | |
QEQSXUNICLDJFE
|
7.3 | IC50 | 2 | — | |
AQSGFRMWBTUZLX
|
7.3 | IC50 | 2 | — | |
XKRJEBDYVJJENF
|
7.3 | IC50 | 2 | — | |
HMHQWJDFNVJCHA
|
7.3 | IC50 | 2 | — | |
SQDVWXKLLQAIME
|
7.3 | IC50 | 2 | — | |
ONWSLHNXFWHTPI
|
7.3 | IC50 | 2 | — | |
VIBKINRBKYEMIO
|
7.3 | IC50 | 2 | — | |
JDRIHSSGXXPQER
|
7.3 | IC50 | 2 | — | |
VGAOCRUUELSAOE
|
7.3 | IC50 | 2 | — | |
CPRWBXAOXHLKLE
|
7.2 | IC50 | 2 | — | |
CTHMWOXOLOMKJN
|
7.2 | IC50 | 2 | — | |
FAKRMULLXOZHQH
|
7.2 | IC50 | 2 | — | |
ITBJNHRCCGGAEF
|
7.2 | IC50 | 2 | — | |
ZDVZBRWEKLWNNU
|
7.2 | IC50 | 2 | — | |
XPAXKCIYJFUWIH
|
7.2 | IC50 | 2 | — | |
PCWGVOYQPPLYQR
|
7.2 | Ki | 2 | — | |
OESBGPUASHCWCC
|
7.2 | IC50 | 2 | — | |
CEDOVDFAPKPYNH
|
7.2 | IC50 | 2 | — | |
HLSAPWPGQUYJIF
|
7.2 | IC50 | 2 | — | |
OWWBGDQUBCMYNV
|
7.1 | IC50 | 2 | — | |
AYTYELJMZUCJQW
|
7.1 | IC50 | 2 | — | |
JJNJJFXIHCARFH
|
7.1 | IC50 | 2 | — | |
CEDOVDFAPKPYNH
|
7.1 | IC50 | 4 | — | |
INRFCWJEFIPMRA
|
7.1 | IC50 | 2 | — | |
KWSSMBHDMXPYIA
|
7.1 | Ki | 2 | — | |
OUVWZPPMRFXVAK
|
7.1 | IC50 | 3 | — | |
WMNWUDVVQXRJTE
|
7.1 | IC50 | 2 | — | |
QYHWCROWSKRSHP
|
7.1 | IC50 | 2 | — | |
WZWYFZNRKHDVOS
|
7.1 | IC50 | 2 | — | |
JCTRAYIUGCXVJI
|
7.1 | IC50 | 2 | — | |
JLTZSOKUYFJVEB
|
7.1 | IC50 | 2 | — | |
SWCZIYPIOLKCKW
|
7.1 | IC50 | 2 | — | |
JKXDDWZJDSDXQN
|
7.0 | IC50 | 2 | — | |
NZEJDWLLYAMAEP
|
7.0 | IC50 | 2 | — | |
PXEGUTANSALZSH
|
7.0 | IC50 | 2 | — | |
UEWSGKREJWLMAB
|
7.0 | IC50 | 2 | — | |
WWQGRJKCRKPKOX
|
7.0 | IC50 | 2 | — | |
BJHIXFJCINNTFW
|
7.0 | IC50 | 2 | — | |
FQGIFVMQXGSXBK
|
7.0 | IC50 | 2 | — | |
OKXUTGCKRRIHII
|
7.0 | IC50 | 2 | — | |
ZXKRUUIFJDOFGA
|
7.0 | IC50 | 2 | — | |
BEZDZMQEVWAVTH
|
7.0 | IC50 | 3 | — | |
BKRYLNPFZBMBFV
|
7.0 | IC50 | 2 | — | |
CLFHIUSNARCPIQ
|
7.0 | IC50 | 2 | — |