Target Details
| UniProt AC | P0AES4 |
|---|---|
| Gene Symbol | gyrA |
| Protein Name | DNA gyrase subunit A |
| Organism | Escherichia coli (strain K12) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF03989 (DNA_gyraseA_C) PF00521 (DNA_topoisoIV) |
Summary
- Multi-target molecules 348
- Clinical molecules 0
- Avg pChEMBL 7.04
Active Molecules (348)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAIGENGZIZRWMW
|
7.9 | IC50 | 2 | — | |
FWKBFPFKHVTISW
|
7.9 | IC50 | 2 | — | |
IPDBXDUZQQUXFU
|
7.9 | IC50 | 2 | — | |
JXMRFLWUZASPFL
|
7.9 | IC50 | 2 | — | |
ZKNZKHAAVPVEAJ
|
7.9 | IC50 | 2 | — | |
GILVJABPOPBFRB
|
7.8 | IC50 | 2 | — | |
NKCCKBBSHMGYMD
|
7.8 | IC50 | 2 | — | |
ADASGIIHCQJGMX
|
7.8 | Ki | 3 | — | |
IIGBANOVZFEHJC
|
7.8 | IC50 | 2 | — | |
XZLCLAKXNCMYKU
|
7.8 | IC50 | 2 | — | |
BYYFORUHJRHMMU
|
7.8 | IC50 | 2 | — | |
BYYFORUHJRHMMU
|
7.8 | IC50 | 2 | — | |
IEHUSEXPEOJDEF
|
7.8 | IC50 | 2 | — | |
YFRGLVPTZHJWIM
|
7.8 | IC50 | 2 | — | |
RLIDZVBFXZCVEH
|
7.8 | IC50 | 2 | — | |
VMFOCQGPXUINDE
|
7.7 | Ki | 3 | — | |
FSOAZMGZMXDGQX
|
7.7 | IC50 | 2 | — | |
VLCKPYIQPLGTCI
|
7.7 | IC50 | 2 | — | |
JNNGDPHORQARNC
|
7.7 | Ki | 2 | — | |
OYTVSJBMPLZYQI
|
7.7 | IC50 | 2 | — | |
VQYUKJQPDIGREC
|
7.7 | IC50 | 2 | — | |
YOFXMMYBDPSZAB
|
7.7 | IC50 | 2 | — | |
LGQLJKHATNDFOW
|
7.7 | IC50 | 2 | — | |
RXANXGVEULKMLY
|
7.7 | IC50 | 3 | — | |
BGZNIXFHOSDNBY
|
7.7 | IC50 | 2 | — | |
AMYYSRVSJKCUAD
|
7.6 | IC50 | 2 | — | |
HKGIQYKOHZBOTG
|
7.6 | IC50 | 2 | — | |
IPDBXDUZQQUXFU
|
7.6 | IC50 | 2 | — | |
YQKWXWMRYFPDSX
|
7.6 | IC50 | 2 | — | |
FWKBFPFKHVTISW
|
7.6 | IC50 | 2 | — | |
HIZAXRZCORUSNT
|
7.6 | IC50 | 2 | — | |
OTIMTRNHWWKMHS
|
7.6 | IC50 | 2 | — | |
REMFYECIOFGXBB
|
7.6 | IC50 | 2 | — | |
IYJZRZIDVYDIHE
|
7.5 | IC50 | 3 | — | |
GAUTWGMJXMALGW
|
7.5 | IC50 | 2 | — | |
QOIXLMNVJYVPLA
|
7.5 | IC50 | 4 | — | |
WNWGHNNOTRTXOM
|
7.5 | IC50 | 2 | — | |
YQKWXWMRYFPDSX
|
7.5 | IC50 | 2 | — | |
QISBQJCTBKCLRU
|
7.5 | IC50 | 2 | — | |
KYOIGEZIXURVNO
|
7.5 | IC50 | 2 | — | |
BZHOCXNKZAJZJC
|
7.5 | Ki | 3 | — | |
OZDLVAWIASMACL
|
7.5 | IC50 | 2 | — | |
UNPWBBYTMMYTPY
|
7.4 | IC50 | 3 | — | |
MHDUFODFABPRAE
|
7.4 | IC50 | 2 | — | |
IPGUFGCGLXUDOJ
|
7.4 | IC50 | 2 | — | |
RVKZOHUACTYRCJ
|
7.4 | IC50 | 2 | — | |
GEDDMFGBKRREEU
|
7.4 | IC50 | 2 | — | |
XKRJEBDYVJJENF
|
7.4 | IC50 | 2 | — | |
YRWGIADUYLSRMK
|
7.4 | IC50 | 2 | — | |
YSAOQGLUGNNBME
|
7.4 | IC50 | 2 | — |