Target Details
| UniProt AC | P0A0K8 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 219
- Clinical molecules 0
- Avg pChEMBL 7.26
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXBBGIQQSYFFLN
|
6.9 | IC50 | 2 | — | |
KWSSMBHDMXPYIA
|
6.9 | Ki | 2 | — | |
RXPOVSSVBGRCOL
|
6.9 | IC50 | 4 | — | |
PVXIXLXRCQEKAV
|
6.8 | IC50 | 2 | — | |
HVMVZISHQKEBLK
|
6.8 | IC50 | 4 | — | |
ASSSIFUQVIZHMH
|
6.8 | IC50 | 4 | — | |
LCOLURQRVPFTDK
|
6.8 | IC50 | 2 | — | |
MTZDGHNXQDFUTD
|
6.8 | IC50 | 2 | — | |
WPELWRSZEWXHNV
|
6.8 | IC50 | 2 | — | |
XMEXMBWRTDMDET
|
6.8 | IC50 | 2 | — | |
IDBNSMFFTLKKMN
|
6.8 | IC50 | 4 | — | |
PZFAZQUREQIODZ
|
6.8 | IC50 | 2 | — | |
ACCKRUPDYNOTMI
|
6.8 | IC50 | 2 | — | |
KTDQGQFRRTZMBJ
|
6.8 | IC50 | 2 | — | |
NHXTWWVJRWMAAW
|
6.7 | IC50 | 4 | — | |
GOMYQMSOGFDKOC
|
6.7 | IC50 | 2 | — | |
PTUWCOMLTLLKMO
|
6.7 | IC50 | 2 | — | |
SIJUCHAWQHDVQI
|
6.7 | Ki | 2 | — | |
USGHRRVFKSLEJT
|
6.7 | IC50 | 4 | — | |
BCOYDHFZZXSZFA
|
6.7 | IC50 | 3 | — | |
JRAGTUWUNIDVFX
|
6.7 | IC50 | 4 | — | |
QUTCIOKBWBLIHI
|
6.7 | IC50 | 2 | — | |
VINPUJZJRCEBET
|
6.7 | IC50 | 5 | — | |
FGJQMRKSDIRTPZ
|
6.6 | IC50 | 2 | — | |
KDGQBAIMBSYHIS
|
6.6 | IC50 | 4 | — | |
CYZXIGIUUJGEAZ
|
6.6 | IC50 | 2 | — | |
OKENRSAOABWGQG
|
6.6 | IC50 | 2 | — | |
HPAZHEGIKZGDCM
|
6.6 | IC50 | 2 | — | |
JCIZDZAGSUATFA
|
6.6 | IC50 | 2 | — | |
QUDWUIDMIRCCRB
|
6.6 | IC50 | 4 | — | |
CHZUNXJHDDAQCN
|
6.5 | IC50 | 2 | — | |
GGBBBGOHXWJLMT
|
6.5 | IC50 | 2 | — | |
XSSZBMPRNHMAKY
|
6.5 | IC50 | 2 | — | |
YOYJNWLSAZAWII
|
6.5 | IC50 | 2 | — | |
MTXGSGLDYXIXFF
|
6.5 | IC50 | 2 | — | |
NJYBFGSBBSLYJT
|
6.5 | IC50 | 2 | — | |
FBPOTAKJJMHABF
|
6.5 | IC50 | 2 | — | |
XSXONJWDSRZBAF
|
6.5 | IC50 | 2 | — | |
NIYHGMQLZAKUHX
|
6.4 | IC50 | 2 | — | |
WAEUAYAUPYCHGQ
|
6.4 | IC50 | 2 | — | |
FMRGAIDONMILDD
|
6.4 | IC50 | 2 | — | |
LSJGLPVZTDCYHQ
|
6.4 | IC50 | 2 | — | |
NAIYBWHMNBAOOG
|
6.4 | IC50 | 2 | — | |
PVQZLFGKXHAYPL
|
6.4 | IC50 | 2 | — | |
ZPMXCTSMZFCELU
|
6.4 | IC50 | 2 | — | |
LTAIYJYCNFSYJU
|
6.4 | IC50 | 2 | — | |
SHKVDXCLBNOXFB
|
6.3 | IC50 | 4 | — | |
FWSHCMNGNALZOS
|
6.3 | IC50 | 2 | — | |
NPQDLAMGUSTRMY
|
6.3 | Ki | 3 | — | |
NVTFDVCDEYDKOF
|
6.3 | IC50 | 2 | — |