Target Details
| UniProt AC | P0A0K8 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 219
- Clinical molecules 0
- Avg pChEMBL 7.26
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NIIWFDOFEHUZBO
|
7.3 | IC50 | 4 | — | |
XQIQPWLZMBMFEZ
|
7.3 | IC50 | 2 | — | |
JNNGDPHORQARNC
|
7.3 | Ki | 2 | — | |
GFQDXSUJWFUHQT
|
7.3 | IC50 | 4 | — | |
BEOSXWIEPVUVCZ
|
7.3 | IC50 | 2 | — | |
COTQDURISRILOR
|
7.3 | IC50 | 2 | — | |
IBUUDJJQWLQLAV
|
7.3 | IC50 | 2 | — | |
FKYJTRSZYAUQIF
|
7.2 | IC50 | 2 | — | |
HGMMQCMKBSYTFD
|
7.2 | IC50 | 2 | — | |
MCUJWFPIOPLDLN
|
7.2 | IC50 | 2 | — | |
UYUKGVMPADBCHE
|
7.2 | IC50 | 2 | — | |
YERDVHADHPXHFF
|
7.2 | IC50 | 4 | — | |
ZFMCWMJGTDHLKI
|
7.2 | IC50 | 4 | — | |
SEAMOYQPPFJZJR
|
7.2 | IC50 | 2 | — | |
VSRUEFVCYYXLCL
|
7.2 | IC50 | 4 | — | |
KLRROQBNYDDGAK
|
7.2 | IC50 | 2 | — | |
NNEBZSDVZCUBGK
|
7.2 | IC50 | 2 | — | |
OWUGLCKBNARAPP
|
7.2 | IC50 | 2 | — | |
MOSDWLNSTVBDPJ
|
7.2 | IC50 | 2 | — | |
OTZGDJFOSDFRBQ
|
7.1 | Ki | 2 | — | |
LHPGCGRDVFMGGQ
|
7.1 | IC50 | 2 | — | |
PCWGVOYQPPLYQR
|
7.1 | Ki | 2 | — | |
JHJANKDCEYKCQY
|
7.0 | IC50 | 4 | — | |
LMBMQPCDCXNUGI
|
7.0 | IC50 | 2 | — | |
PNXMNHGKWCLCMU
|
7.0 | IC50 | 4 | — | |
WMNKVDSSYPIFBR
|
7.0 | IC50 | 2 | — | |
PQWWHNZAZANFOZ
|
7.0 | IC50 | 5 | — | |
CZTMTIJJNWLREO
|
7.0 | IC50 | 2 | — | |
RSJIYODUVAGVDD
|
7.0 | IC50 | 2 | — | |
MCMNYTOHUPZLOA
|
6.9 | IC50 | 5 | — | |
IYDSEXALBFJDID
|
6.9 | IC50 | 2 | — | |
BMANDSXMIVZGEY
|
6.9 | IC50 | 2 | — | |
KFEYIAJIUJJIRU
|
6.9 | IC50 | 2 | — | |
AUXHQPYDIVPJQT
|
6.9 | IC50 | 2 | — | |
DNYLEYUAAXOKIE
|
6.9 | IC50 | 2 | — | |
FBUOCINPAWXYMK
|
6.9 | IC50 | 2 | — | |
GUEBWQFTJDQZMH
|
6.9 | IC50 | 2 | — | |
HDUOQGPJPLEPTI
|
6.9 | IC50 | 2 | — | |
IGGQZENFMDGPEU
|
6.9 | IC50 | 2 | — | |
NDXWAAKFUDDIDP
|
6.9 | IC50 | 2 | — | |
OCZXFLPYVJPVBO
|
6.9 | IC50 | 2 | — | |
PEKRPORMYGTOHQ
|
6.9 | IC50 | 4 | — | |
ROYGGNJCSVBHRS
|
6.9 | IC50 | 2 | — | |
RXUHYHMLLDSVIR
|
6.9 | IC50 | 2 | — | |
STJYMKNNSABJJZ
|
6.9 | IC50 | 2 | — | |
STVLAIOEZXTGBZ
|
6.9 | IC50 | 2 | — | |
VQIOYVHLFZXJKX
|
6.9 | IC50 | 2 | — | |
VRARNXIVPHOALP
|
6.9 | IC50 | 2 | — | |
WCUIUMSVLSFGOF
|
6.9 | IC50 | 2 | — | |
WTWWYEPNQHNZPG
|
6.9 | IC50 | 2 | — |