Target Details
| UniProt AC | P0A0K8 |
|---|---|
| Gene Symbol | gyrB |
| Protein Name | DNA gyrase subunit B |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00204 (DNA_gyraseB) PF00986 (DNA_gyraseB_C) PF02518 (HATPase_c) PF01751 (Toprim) |
Summary
- Multi-target molecules 219
- Clinical molecules 0
- Avg pChEMBL 7.26
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZKUQOZGHQRJHO
|
8.9 | IC50 | 2 | — | |
XMRMYIYEEWALOZ
|
8.9 | IC50 | 4 | — | |
ALUMFQDCLSGUTJ
|
8.7 | IC50 | 2 | — | |
FNBRRJMBTVMTJT
|
8.7 | IC50 | 2 | — | |
JPHRWMIBMBVHII
|
8.7 | IC50 | 2 | — | |
QTISQBZFCNUZBT
|
8.7 | IC50 | 2 | — | |
UEONWFOAVQSBSL
|
8.7 | IC50 | 2 | — | |
VGUDXZMFJGEQIG
|
8.7 | IC50 | 2 | — | |
ZZNKKJQEANOWCQ
|
8.7 | IC50 | 2 | — | |
VDEMYFZESGTBQM
|
8.6 | IC50 | 2 | — | |
DYFJTHKGNCSRJG
|
8.5 | IC50 | 2 | — | |
BGDGHNSKANYMHF
|
8.4 | IC50 | 2 | — | |
QMBIGGCLOHYBHN
|
8.4 | IC50 | 4 | — | |
RDTDFCZCBIXFEI
|
8.4 | IC50 | 5 | — | |
WTIJXIZOODAMJT
|
8.2 | IC50 | 2 | — | |
IXXRRXMYIMRHHE
|
8.2 | Ki | 3 | — | |
QWDBLAFTHZKKSX
|
8.1 | IC50 | 2 | — | |
BMGHOFGNTZXSPS
|
8.1 | IC50 | 2 | — | |
CEDOAZZFPILAKJ
|
8.1 | IC50 | 2 | — | |
CRZVOEIRSRPIPL
|
8.1 | IC50 | 2 | — | |
CSUATDQKJHRXBT
|
8.1 | IC50 | 2 | — | |
GIYAXUINNMNECB
|
8.1 | IC50 | 2 | — | |
IECLISBCGWXBCN
|
8.1 | IC50 | 2 | — | |
IHEDUPSAYQMLJB
|
8.1 | IC50 | 2 | — | |
KYHZWYOJTBVISH
|
8.1 | IC50 | 2 | — | |
KYHZWYOJTBVISH
|
8.1 | IC50 | 2 | — | |
LSLCINNAJSZAFZ
|
8.1 | IC50 | 2 | — | |
OWUDSPGWMNOZFU
|
8.1 | Ki | 3 | — | |
PUJSFHKEPIXRAF
|
8.1 | IC50 | 2 | — | |
QCXZBOAXZXYRAD
|
8.1 | IC50 | 2 | — | |
SPSUUIZYXVETJI
|
8.1 | IC50 | 2 | — | |
SUUQDWDDUCAXHF
|
8.1 | IC50 | 2 | — | |
USABNRUSMYNPRU
|
8.1 | IC50 | 2 | — | |
XSEHYVUOJSOPPX
|
8.1 | IC50 | 2 | — | |
YRUUNFHQHJGHTP
|
8.1 | IC50 | 2 | — | |
YZUZZSIWAUWQQQ
|
8.1 | IC50 | 2 | — | |
ZQYNHBTULYYGMD
|
8.1 | IC50 | 2 | — | |
BKUISYCLLXCBJV
|
8.1 | Ki | 4 | — | |
IKNUYGJLHHAVHT
|
8.1 | IC50 | 2 | — | |
NTNKQRBKOGURQE
|
8.1 | IC50 | 4 | — | |
YQTBDIINFUTVKB
|
8.0 | IC50 | 2 | — | |
FNBRRJMBTVMTJT
|
8.0 | IC50 | 2 | — | |
ULFIHHOZULSWER
|
8.0 | Ki | 3 | — | |
YVYGZNXCUWXRQN
|
8.0 | Ki | 3 | — | |
XTMGTPTXHXWURI
|
7.9 | Ki | 3 | — | |
REEOSLJMDKKLQA
|
7.9 | IC50 | 4 | — | |
GJIJCAIHXYJAQJ
|
7.8 | IC50 | 2 | — | |
NKXJSCXEAVZSMF
|
7.8 | IC50 | 3 | — | |
ZAVBNYFZECWAQQ
|
7.8 | IC50 | 2 | — | |
DIIRMLRBGBCXMK
|
7.8 | Ki | 3 | — |