Target Details
| UniProt AC | P0A017 |
|---|---|
| Gene Symbol | folA |
| Protein Name | Dihydrofolate reductase |
| Organism | Staphylococcus aureus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 96
- Clinical molecules 0
- Avg pChEMBL 8.88
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KDNYRYCRFHVZNX
|
8.8 | Ki | 2 | — | |
RHPGXKNMHAITAC
|
8.8 | Ki | 2 | — | |
HWJPWWYTGBZDEG
|
8.7 | IC50 | 2 | — | |
LBQMRSNKEUNXMT
|
8.6 | IC50 | 4 | — | |
HWJPWWYTGBZDEG
|
8.6 | IC50 | 2 | — | |
JTOMSJOIFXSANF
|
8.6 | Ki | 2 | — | |
VDZFKJHFXFCADG
|
8.6 | Ki | 2 | — | |
YGDVMSPWZQHNMB
|
8.5 | IC50 | 2 | — | |
YUQSMDFWZIVXAK
|
8.5 | Ki | 2 | — | |
MDBNODWEXWKOIX
|
8.5 | Ki | 2 | — | |
IFLADHLPWSCQJK
|
8.4 | Ki | 2 | — | |
BGVUMMFSZABYHW
|
8.4 | Ki | 2 | — | |
NNGNWTVCPVJZTD
|
8.3 | Ki | 2 | — | |
VQOBXMVKFHMZJP
|
8.0 | Ki | 2 | — | |
NQHZOWBSMCFILX
|
8.0 | IC50 | 4 | — | |
COHGVYNMDPBQFR
|
7.9 | IC50 | 3 | — | |
GCDLAOPKRFVDHQ
|
7.9 | Ki | 4 | — | |
KEPLBUUTAQCZOE
|
7.8 | Ki | 3 | — | |
PPKWGSTVAQFAGZ
|
7.8 | Ki | 2 | — | |
NQHZOWBSMCFILX
|
7.8 | IC50 | 4 | — | |
NQHZOWBSMCFILX
|
7.7 | IC50 | 4 | — | |
KEPLBUUTAQCZOE
|
7.7 | Ki | 3 | — | |
LMFGVRPNYCLJOJ
|
7.7 | IC50 | 3 | — | |
CZCHMGRCEXJPTP
|
7.7 | IC50 | 3 | — | |
GNXVOAVSOLSRGY
|
7.6 | IC50 | 3 | — | |
DNZHKQMESCYJCG
|
7.6 | IC50 | 3 | — | |
DNZHKQMESCYJCG
|
7.6 | IC50 | 3 | — | |
ULSWBNKDTMSHNY
|
7.6 | IC50 | 3 | — | |
DGJGWMFHVPDAKM
|
7.5 | IC50 | 4 | — | |
JQPNVLABZWBWEL
|
7.5 | IC50 | 4 | — | |
AATPYXMXFBBKFO
|
7.5 | IC50 | 3 | — | |
IXYIZEGMHCDBOH
|
7.5 | IC50 | 3 | — | |
UEZKDWYIIOOENX
|
7.5 | IC50 | 3 | — | |
ATFDKOLABYIYCC
|
7.4 | IC50 | 4 | — | |
ATFDKOLABYIYCC
|
7.4 | IC50 | 4 | — | |
BYYHQKXHHYWFBF
|
7.4 | IC50 | 2 | — | |
QKLZHVMWTSBUFL
|
7.2 | IC50 | 4 | — | |
JPENSYBRTSIYGO
|
7.2 | IC50 | 3 | — | |
JPENSYBRTSIYGO
|
7.2 | IC50 | 5 | — | |
NUZPENCTXJLJCY
|
7.2 | IC50 | 2 | — | |
FHTSRDNJZWDVBC
|
7.2 | IC50 | 3 | — | |
IDRYQRLCJXCFLM
|
7.1 | IC50 | 2 | — | |
PFZXPVFWXCUAJW
|
7.1 | IC50 | 4 | — | |
NNFDQABYXZBKRK
|
6.7 | IC50 | 4 | — | |
QVXYJVHNRPNRJL
|
6.4 | IC50 | 3 | — | |
QVXYJVHNRPNRJL
|
6.4 | IC50 | 3 | — |