Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OLJYGSVADWZNIQ
|
8.1 | IC50 | 2 | — | |
UEVFMGJBRLJVKO
|
8.1 | IC50 | 3 | — | |
FBGYDRBIQYAULP
|
8.1 | IC50 | 2 | — | |
FSFKDNPHPFINJD
|
8.1 | IC50 | 3 | — | |
LVZZNRAHJDTKAL
|
8.1 | IC50 | 2 | — | |
PCHKPVIQAHNQLW
|
8.1 | IC50 | 8 | — | |
DBTLGWQFPVIXTJ
|
8.1 | IC50 | 2 | — | |
GXLCEYYXBWDRJO
|
8.1 | IC50 | 3 | — | |
RZVRCAKYGAURIU
|
8.1 | IC50 | 2 | — | |
GFUWRTZMZMICED
|
8.1 | IC50 | 3 | — | |
JHSRPZWVYSMIQK
|
8.1 | IC50 | 2 | — | |
ZMBBXGKYRZNGTQ
|
8.1 | IC50 | 2 | — | |
DWPOZLNCERCETA
|
8.1 | IC50 | 2 | — | |
FLTKNCUXYGRLOI
|
8.1 | IC50 | 2 | — | |
HTMPMXJFMOUCOQ
|
8.1 | IC50 | 2 | — | |
QAJSMIVRRQDYBG
|
8.1 | IC50 | 3 | — | |
SJFGTXAAKCLIOI
|
8.1 | IC50 | 2 | — | |
YLXGAIYNRGPZSR
|
8.1 | IC50 | 2 | — | |
CKCMEFFRRGTNSY
|
8.0 | IC50 | 2 | — | |
IRVJFMHHDJQNGA
|
8.0 | IC50 | 2 | — | |
RYCVFUGCROLXMH
|
8.0 | IC50 | 2 | — | |
SOASXIFPFLUWRH
|
8.0 | IC50 | 2 | — | |
XDQDKCGQZXCZGC
|
8.0 | IC50 | 2 | — | |
AFXJUCILCGBUNX
|
8.0 | IC50 | 4 | — | |
AMWNTQXPBJQZET
|
8.0 | IC50 | 3 | — | |
FHQJOMRJKRMAOH
|
8.0 | IC50 | 2 | — | |
QEEHFLKQODURKT
|
8.0 | IC50 | 2 | — | |
QSDUGBPLSHIMHQ
|
8.0 | IC50 | 3 | — | |
SMSCYHHVBZIUMV
|
8.0 | IC50 | 2 | — | |
SRPQZLVMAZBVEH
|
8.0 | IC50 | 2 | — | |
SUFHZCQTMDLDRK
|
8.0 | IC50 | 2 | — | |
WNMYZOLGAGNXGE
|
8.0 | IC50 | 2 | — | |
XVWZUMYLDUPVRN
|
8.0 | IC50 | 2 | — | |
GGJVOTFHPYZESL
|
8.0 | IC50 | 4 | — | |
GSHBUCNCWYHWKA
|
8.0 | IC50 | 2 | — | |
IRZDTZKFGZNLMK
|
8.0 | IC50 | 2 | — | |
IZPURWNXWPTMHH
|
8.0 | IC50 | 2 | — | |
JHHJWGJMKVRLMC
|
8.0 | IC50 | 2 | — | |
KVSHPARHGQSONL
|
8.0 | IC50 | 2 | — | |
PQFMYQNBODJBRE
|
8.0 | Ki | 2 | — | |
RCNMQXVWWXSESA
|
8.0 | IC50 | 3 | — | |
VUECMVWDRZENTP
|
8.0 | Kd | 2 | — | |
SOASXIFPFLUWRH
|
8.0 | IC50 | 3 | — | |
CEGOEVTXZXXUSN
|
8.0 | IC50 | 2 | — | |
PMIVWECZXHTRTB
|
8.0 | IC50 | 2 | — | |
ASIFNLNMOYRKGY
|
8.0 | IC50 | 2 | — | |
DXBJWAWQZDLDNB
|
8.0 | IC50 | 2 | — | |
HTRPLWGQNMXGRD
|
8.0 | IC50 | 3 | — | |
NLVNPTRNTQDKPQ
|
8.0 | IC50 | 2 | — | |
VAOQBNBDBKHNQY
|
8.0 | IC50 | 3 | — |