Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UOAHTPZUUUBPBK
|
8.2 | IC50 | 3 | — | |
ZMNGPSRBNIMINA
|
8.2 | IC50 | 2 | — | |
ZMRSDMLCFJDLKR
|
8.2 | IC50 | 3 | — | |
FLCHMGRFSJQORK
|
8.2 | IC50 | 3 | — | |
BJFLQGUKMCVUMZ
|
8.2 | IC50 | 2 | — | |
MFPOWTKEAYCCGQ
|
8.2 | IC50 | 2 | — | |
QCDZWDMYQRCVLA
|
8.2 | IC50 | 2 | — | |
ANXRWJLGPPKOSD
|
8.2 | IC50 | 2 | — | |
BSHNSNFEEYZSMQ
|
8.2 | IC50 | 2 | — | |
CCWTWPIDXUGAKX
|
8.2 | IC50 | 3 | — | |
DEPHVBQJDPPGQN
|
8.2 | IC50 | 2 | — | |
DETVQHYFSHWWBS
|
8.2 | IC50 | 2 | — | |
HGEPGGJUGUMFHT
|
8.2 | IC50 | 2 | — | |
JKCHNICKXRIXAL
|
8.2 | IC50 | 2 | — | |
KJYNUBQNUKNDSF
|
8.2 | IC50 | 2 | — | |
NIOMTPKIOLNRTQ
|
8.2 | IC50 | 2 | — | |
NJQTWWNECKEAQJ
|
8.2 | IC50 | 3 | — | |
PITKHMJQSBHPED
|
8.2 | IC50 | 3 | — | |
PZDZBZWWQUDTKX
|
8.2 | IC50 | 3 | — | |
SCONNUWWGIRXAF
|
8.2 | IC50 | 2 | — | |
UGDXZOURHPLYNW
|
8.2 | Ki | 2 | — | |
UWHPKMURHNFAOY
|
8.2 | IC50 | 2 | — | |
ZXSZFRRHHIPVGQ
|
8.2 | IC50 | 2 | — | |
AURCLDMUVVKGCY
|
8.1 | IC50 | 3 | — | |
MWIUPFYRAAIUMB
|
8.1 | IC50 | 3 | — | |
NBUIWUDKADDAKC
|
8.1 | IC50 | 2 | — | |
QFZBUSJLFWEDKO
|
8.1 | IC50 | 2 | — | |
XULZRMKGTVQSFV
|
8.1 | IC50 | 2 | — | |
ZGMGCVMYDSXGAA
|
8.1 | IC50 | 2 | — | |
FADNVFGOLBDUSB
|
8.1 | IC50 | 2 | — | |
QWQRHMZFZSWUOD
|
8.1 | IC50 | 3 | — | |
RSZFCUWJGDNCGK
|
8.1 | IC50 | 3 | — | |
TWZQEBQCXWLACN
|
8.1 | IC50 | 3 | — | |
WEFPHDYTHUNVAM
|
8.1 | IC50 | 3 | — | |
DVBFHLPDOMIKKR
|
8.1 | IC50 | 3 | — | |
DXFARVNRLJXDDA
|
8.1 | IC50 | 2 | — | |
JKAHAAKUCDSUBE
|
8.1 | IC50 | 2 | — | |
LGFTWORQFUMEPZ
|
8.1 | IC50 | 2 | — | |
MLYYYJSVHUVZHH
|
8.1 | IC50 | 3 | — | |
NZDMYHLPDHCLGC
|
8.1 | IC50 | 3 | — | |
ORSBXGBOZDSEJT
|
8.1 | IC50 | 3 | — | |
XQOHUNRPGOTXDR
|
8.1 | IC50 | 3 | — | |
CDELRUCHGDJWNM
|
8.1 | IC50 | 3 | — | |
DILZMEVBCHRKIZ
|
8.1 | IC50 | 3 | — | |
FKYXYTRRMYNSQO
|
8.1 | Ki | 2 | — | |
IAOPKPFMQJOUNF
|
8.1 | IC50 | 2 | — | |
JDXLMISSSMZOIL
|
8.1 | IC50 | 2 | — | |
JZCAEMQAGFOICW
|
8.1 | IC50 | 2 | — | |
KXSIHXHEHABEJX
|
8.1 | Ki | 2 | — | |
MZAAUJMUTYAMFB
|
8.1 | IC50 | 2 | — |