Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XPCCVBMKWOBTFC
|
8.3 | IC50 | 2 | — | |
AXXNBSKROWNMJJ
|
8.2 | IC50 | 2 | — | |
LRRAZXKYVVVMLY
|
8.2 | IC50 | 2 | — | |
SOASXIFPFLUWRH
|
8.2 | IC50 | 2 | — | |
HGJVONCBQFKWRI
|
8.2 | IC50 | 2 | — | |
IXTIMUQTDOPTKU
|
8.2 | IC50 | 2 | — | |
IZSILESJFBWTKL
|
8.2 | IC50 | 2 | — | |
LZMKLHYIPIJTRL
|
8.2 | IC50 | 2 | — | |
POZQILOZTPZMDN
|
8.2 | IC50 | 2 | — | |
AHZFXBYDJSLSCQ
|
8.2 | IC50 | 2 | — | |
XGFMLKJENFANEN
|
8.2 | IC50 | 2 | — | |
ZGDNFPWQEQSQAA
|
8.2 | IC50 | 3 | — | |
DXTVYXKOSJALKU
|
8.2 | IC50 | 2 | — | |
FHXVYSAVWVGYSB
|
8.2 | IC50 | 2 | — | |
FPMIUVGZAHMUQO
|
8.2 | IC50 | 2 | — | |
GFHLWWHOLUWZLZ
|
8.2 | IC50 | 4 | — | |
GYNGGIICQNEJEN
|
8.2 | IC50 | 2 | — | |
HETQFLWNGHJHJZ
|
8.2 | IC50 | 2 | — | |
IWIRGSJMTCVGQQ
|
8.2 | IC50 | 2 | — | |
LGVIXHMVSRYWJL
|
8.2 | Ki | 2 | — | |
NVYAWMBGKKEULL
|
8.2 | IC50 | 2 | — | |
ORFAAEFWFKRACI
|
8.2 | IC50 | 2 | — | |
OUERNEXEYTUWRZ
|
8.2 | IC50 | 3 | — | |
QYDURWHTEIUTEI
|
8.2 | IC50 | 4 | — | |
RRMZVMRBJRDAFX
|
8.2 | Ki | 2 | — | |
WELSPTLZWKCYMB
|
8.2 | IC50 | 3 | — | |
YBQAXMUUMRZOKE
|
8.2 | IC50 | 2 | — | |
YKIBUJVDRWECHV
|
8.2 | IC50 | 3 | — | |
ZBCWPRMBUXOZEF
|
8.2 | Ki | 2 | — | |
BJFLQGUKMCVUMZ
|
8.2 | IC50 | 2 | — | |
CDFHCXNQPYQRFI
|
8.2 | IC50 | 2 | — | |
RGEGQSNDVNAPBM
|
8.2 | IC50 | 2 | — | |
TWNKKSWDODFPFW
|
8.2 | IC50 | 2 | — | |
UYHSCMQSBJXZGX
|
8.2 | IC50 | 4 | — | |
YTZCTEISEKPJTQ
|
8.2 | IC50 | 3 | — | |
BDGRZWISYNXFKD
|
8.2 | IC50 | 3 | — | |
DBLBOZLZPCJKAH
|
8.2 | IC50 | 3 | — | |
HHHFTURDICHXNW
|
8.2 | IC50 | 3 | — | |
JFJGQBKALIOSDA
|
8.2 | IC50 | 3 | — | |
QBLCDAXXROYNNC
|
8.2 | IC50 | 2 | — | |
AHDIVRNRWIUPJX
|
8.2 | IC50 | 3 | — | |
HPAHIIGPVDRZLN
|
8.2 | IC50 | 2 | — | |
KOMGSVVWXUEBNT
|
8.2 | IC50 | 3 | — | |
LIYLVRUTQRQGPO
|
8.2 | IC50 | 2 | — | |
SVYQAPDHJLXDGC
|
8.2 | IC50 | 3 | — | |
CINNRILLZCDNOZ
|
8.2 | IC50 | 3 | — | |
GXXRJPKTTBCLNF
|
8.2 | IC50 | 2 | — | |
INRRUWSEBDJLPW
|
8.2 | IC50 | 3 | — | |
PVOOFJMJDHPMBT
|
8.2 | IC50 | 2 | — | |
SJYGJUQORXZRIJ
|
8.2 | IC50 | 3 | — |