Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BLZYPQSTOPUZPW
|
8.4 | IC50 | 2 | — | |
MKWJWRCMHZZWAU
|
8.4 | IC50 | 2 | — | |
XBHZTKNYGUXRMG
|
8.4 | IC50 | 2 | — | |
YCMALEKADPQGHA
|
8.4 | IC50 | 2 | — | |
CEUSZBDWOAZEBV
|
8.4 | IC50 | 2 | — | |
DQGBARZZIIDDAZ
|
8.3 | IC50 | 2 | — | |
FBIGNDFZRCUSDQ
|
8.3 | IC50 | 3 | — | |
GBEWXEQDDXPZJQ
|
8.3 | IC50 | 2 | — | |
IFGWKNJRNNUOIA
|
8.3 | IC50 | 2 | — | |
LDUXKZCPPPHDPU
|
8.3 | IC50 | 2 | — | |
ONEIDYKHPRMDQO
|
8.3 | IC50 | 3 | — | |
VQGIUGREGZOJMG
|
8.3 | IC50 | 2 | — | |
BJIIXHJAFPCRRA
|
8.3 | IC50 | 2 | — | |
NRDDMPIVXPOIMZ
|
8.3 | IC50 | 2 | — | |
QBWWPFIBJGBBKX
|
8.3 | IC50 | 2 | — | |
UTWLDWAFEKZNCC
|
8.3 | IC50 | 2 | — | |
ZIZAGKWTJFKACS
|
8.3 | IC50 | 2 | — | |
CVTFVYCHNGODLR
|
8.3 | IC50 | 3 | — | |
FJOFREJOLJFMNF
|
8.3 | IC50 | 3 | — | |
OCLDJPYPPFDDNO
|
8.3 | IC50 | 3 | — | |
WPSFTNDXYZENJA
|
8.3 | IC50 | 3 | — | |
ADAAOWJCZJSQAB
|
8.3 | IC50 | 2 | — | |
DPKCTDXZHPAPLS
|
8.3 | IC50 | 3 | — | |
ICWAHMDHBIKSJI
|
8.3 | IC50 | 2 | — | |
KXXRGTYOVUETBV
|
8.3 | IC50 | 3 | — | |
VREYQMOSHXUIOX
|
8.3 | IC50 | 2 | — | |
XCULREABYDORQQ
|
8.3 | IC50 | 2 | — | |
AFWLAWBSENRTOI
|
8.3 | IC50 | 2 | — | |
BRHAGWRGTMVKQA
|
8.3 | IC50 | 2 | — | |
DCSUGHIXMFUMOQ
|
8.3 | IC50 | 3 | — | |
FDLYAMZZIXQODN
|
8.3 | IC50 | 11 | — | |
FOGFSNYHDLKAID
|
8.3 | Ki | 2 | — | |
IZKKJBVPFFOLOL
|
8.3 | IC50 | 2 | — | |
JNAHVYVRKWKWKQ
|
8.3 | Ki | 2 | — | |
OAFQCDJUMPFXNS
|
8.3 | IC50 | 2 | — | |
OSCYHTCDAZYCLV
|
8.3 | Ki | 2 | — | |
PQHSBQMZINJNST
|
8.3 | IC50 | 2 | — | |
SYOHFHPKBUPMJS
|
8.3 | IC50 | 3 | — | |
JNAHVYVRKWKWKQ
|
8.3 | IC50 | 4 | — | |
RDWMOYFDWSZBAZ
|
8.3 | IC50 | 3 | — | |
MHQFEYXRRZRKBA
|
8.3 | IC50 | 3 | — | |
RAPGQTWOPCNSEJ
|
8.3 | IC50 | 3 | — | |
UCDKHNXJMSHBER
|
8.3 | IC50 | 2 | — | |
YJBHZZJZTYUYSR
|
8.3 | IC50 | 2 | — | |
BWTOWBOMDHKCDB
|
8.3 | IC50 | 7 | — | |
ONWFSNLHAZAPLW
|
8.3 | IC50 | 3 | — | |
LIQDGVXNWJAUNO
|
8.3 | IC50 | 6 | — | |
MGFDCSFBWGIIJD
|
8.3 | IC50 | 2 | — | |
MZLDTLJZDXBQCV
|
8.3 | IC50 | 2 | — | |
UCQAPUVIUAYEGE
|
8.3 | IC50 | 3 | — |