Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHWBVGUNUQRUHT
|
8.5 | IC50 | 2 | — | |
DJSXTFVMGSHIQP
|
8.5 | IC50 | 2 | — | |
DQGBARZZIIDDAZ
|
8.5 | IC50 | 2 | — | |
IULLGBUVNORARL
|
8.5 | Ki | 2 | — | |
IXNZYKNOAINDTN
|
8.5 | IC50 | 3 | — | |
RJIYGYHNEKRSTG
|
8.5 | Ki | 2 | — | |
UPTYBPOYVNYQMT
|
8.5 | IC50 | 7 | — | |
VXKAXDSVEXWYFC
|
8.5 | IC50 | 2 | — | |
VXYSCPNHOZCHHO
|
8.5 | IC50 | 2 | — | |
WBSPNPVOFBRUKC
|
8.5 | Ki | 2 | — | |
WQAVGRAETZEADU
|
8.5 | IC50 | 2 | — | |
WTKBXXGVXWHMHX
|
8.5 | IC50 | 2 | — | |
YDYWCKXGGCVENO
|
8.5 | IC50 | 2 | — | |
CRTCKATZPLYUCW
|
8.5 | IC50 | 2 | — | |
LLBQUOHKCAYWBR
|
8.5 | IC50 | 2 | — | |
DRPXVULWOOOZDV
|
8.5 | IC50 | 3 | — | |
ROBJKLPZIPNAMV
|
8.5 | IC50 | 2 | — | |
CVLCVUYBIPUQBG
|
8.5 | IC50 | 3 | — | |
DSRLEZVTVWWOOC
|
8.5 | IC50 | 2 | — | |
ISQUAVJORRNWGA
|
8.5 | IC50 | 3 | — | |
OGMWSRSCJFPYFR
|
8.5 | IC50 | 2 | — | |
QJKRRPUDVWORKT
|
8.5 | IC50 | 2 | — | |
UFCYAFSJOZTJKT
|
8.5 | IC50 | 3 | — | |
FWWPLYZVUBCMHN
|
8.5 | IC50 | 2 | — | |
RLKUZCOFKFUEHH
|
8.5 | IC50 | 3 | — | |
YEEMANFJIXWISV
|
8.5 | IC50 | 2 | — | |
HDOXYDHZDFTFMX
|
8.4 | IC50 | 2 | — | |
PZYRHYWULWFGBG
|
8.4 | IC50 | 3 | — | |
XUFWBGKENCGHSD
|
8.4 | IC50 | 3 | — | |
NQEBXSGIXPJSTM
|
8.4 | IC50 | 2 | — | |
XRRMNZJUZRPHGN
|
8.4 | IC50 | 2 | — | |
NTYRAXKJQKLKLY
|
8.4 | IC50 | 2 | — | |
VXXHFHBGNMSWMO
|
8.4 | IC50 | 2 | — | |
MWUSNBQNIIMQRN
|
8.4 | IC50 | 4 | — | |
OXULFDKDMPHAFP
|
8.4 | IC50 | 3 | — | |
WKXCQZQWHUTWSY
|
8.4 | IC50 | 2 | — | |
JQJGYBASPJXNIJ
|
8.4 | IC50 | 3 | — | |
JSGRLNJKTKDILH
|
8.4 | Ki | 2 | — | |
LXMVOWGBBQUTCO
|
8.4 | IC50 | 2 | — | |
PWESUKOHBQOSBW
|
8.4 | Ki | 2 | — | |
RJRQJZUWLRXDTF
|
8.4 | Ki | 2 | — | |
YBQAXMUUMRZOKE
|
8.4 | IC50 | 2 | — | |
ZLFRATDTTALTRO
|
8.4 | Ki | 2 | — | |
PVOOFJMJDHPMBT
|
8.4 | IC50 | 2 | — | |
UAVGSHVHWKPCPP
|
8.4 | IC50 | 3 | — | |
WAODZKSACVYCRN
|
8.4 | IC50 | 20 | — | |
ZOFBQDSFQVONQL
|
8.4 | IC50 | 2 | — | |
ATDFXALCNPKLOR
|
8.4 | IC50 | 2 | — | |
HNUBZGFNRGYRML
|
8.4 | IC50 | 2 | — | |
WVGLSASLDWFLFS
|
8.4 | IC50 | 2 | — |