Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RTNLYODALOPJJQ
|
8.7 | IC50 | 2 | — | |
RVKIODKELWOUEW
|
8.7 | IC50 | 2 | — | |
MBHKTNPQYPMZCA
|
8.7 | IC50 | 2 | — | |
FJMYVHKWFNIERC
|
8.7 | Ki | 2 | — | |
FRTYCOFZECQXQT
|
8.7 | IC50 | 2 | — | |
FRTYCOFZECQXQT
|
8.7 | IC50 | 2 | — | |
FRTYCOFZECQXQT
|
8.7 | IC50 | 2 | — | |
GTBYWKYWQWSPTR
|
8.7 | Ki | 2 | — | |
IXVYIQVZFUMBEX
|
8.7 | IC50 | 2 | — | |
JLFSBHQQXIAQEC
|
8.7 | IC50 | 4 | — | |
JMPOHTPVCKISQL
|
8.7 | IC50 | 3 | — | |
LZXFKOUZJFPYDT
|
8.7 | IC50 | 2 | — | |
NQLKZEKCIROGCB
|
8.7 | IC50 | 2 | — | |
TVOBRCWLURXJSE
|
8.7 | IC50 | 2 | — | |
TYXRAPFGHJZSQQ
|
8.7 | IC50 | 2 | — | |
TYXRAPFGHJZSQQ
|
8.7 | IC50 | 2 | — | |
TYXRAPFGHJZSQQ
|
8.7 | IC50 | 2 | — | |
WARUZPFHLRLCHE
|
8.7 | IC50 | 7 | — | |
HDJIYQABLDDLST
|
8.7 | IC50 | 20 | — | |
POPCEFBMGMRZJG
|
8.7 | IC50 | 2 | — | |
QAYXPOVVNWSHEE
|
8.7 | IC50 | 2 | — | |
YYUSEXNQXFAVSQ
|
8.7 | IC50 | 2 | — | |
FBFODWQRNOVLGQ
|
8.7 | IC50 | 2 | — | |
HBJRTNJBCUCSST
|
8.7 | IC50 | 2 | — | |
NTLIPIHZQJVWJM
|
8.6 | IC50 | 2 | — | |
GRPXLKXGJAGYSD
|
8.6 | IC50 | 3 | — | |
GVVGCLUTJOAUON
|
8.6 | IC50 | 2 | — | |
HYNBNUYQTQIHJK
|
8.6 | IC50 | 2 | — | |
KCBVLLQJPRAPJT
|
8.6 | IC50 | 2 | — | |
XMLOXTGVMSYKHN
|
8.6 | IC50 | 2 | — | |
BOKCRBOZYPDNIC
|
8.6 | IC50 | 3 | — | |
FICCKZPDRHVIJH
|
8.6 | IC50 | 2 | — | |
AGYRIAKSKBQPQX
|
8.6 | IC50 | 2 | — | |
LFYTWGBFZMCREV
|
8.6 | IC50 | 2 | — | |
PHXCOCKVZBWRCP
|
8.6 | IC50 | 2 | — | |
SNSYYJLSJTUZMP
|
8.6 | Ki | 2 | — | |
UYSWVENMUWDLDZ
|
8.6 | IC50 | 2 | — | |
WPTNASIDXWQCDG
|
8.6 | IC50 | 3 | — | |
GXXMDTMOEKZYDT
|
8.6 | IC50 | 2 | — | |
DLDYOMRJCIUSIG
|
8.6 | IC50 | 2 | — | |
FFDCUOYHHZSVET
|
8.6 | IC50 | 2 | — | |
LRRSQDMHWPHEMQ
|
8.6 | IC50 | 2 | — | |
PYDVJBPGFWXTDE
|
8.6 | IC50 | 2 | — | |
CDFHCXNQPYQRFI
|
8.6 | IC50 | 2 | — | |
XKSQRLIEJSXRFK
|
8.6 | IC50 | 2 | — | |
HEDHFDLLWZBOLO
|
8.5 | IC50 | 2 | — | |
LNWPRZVIPZXIHL
|
8.5 | IC50 | 3 | — | |
SDTRERMWZQTLRS
|
8.5 | IC50 | 2 | — | |
QADXMHHSBCIXIC
|
8.5 | IC50 | 2 | — | |
AHIVQGOUBLVTCB
|
8.5 | Ki | 2 | — |