Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHTFNTYBBURGHS
|
9.0 | IC50 | 2 | — | |
NLWYFXIKIPVWHJ
|
9.0 | IC50 | 2 | — | |
OQXRCISZYORQBS
|
9.0 | IC50 | 2 | — | |
PQHSBQMZINJNST
|
9.0 | IC50 | 2 | — | |
QKZGOZNDFYDQOV
|
9.0 | IC50 | 2 | — | |
ZDDPBFWHZOJFHF
|
9.0 | IC50 | 6 | — | |
HUQDBDMQKROGGR
|
9.0 | IC50 | 2 | — | |
GBLMKEGSKITKAH
|
9.0 | IC50 | 2 | — | |
VKMZDQDDIAQHOC
|
9.0 | IC50 | 2 | — | |
IBBZXRLLZKUNIM
|
9.0 | IC50 | 4 | — | |
LVUBLVHQRWQIFH
|
9.0 | IC50 | 2 | — | |
PVOOFJMJDHPMBT
|
9.0 | IC50 | 2 | — | |
PZDZBMUDLPDHQV
|
9.0 | IC50 | 2 | — | |
RKOUKZKFCAOXCG
|
9.0 | IC50 | 2 | — | |
JFZQZMDWGYRERP
|
8.9 | IC50 | 3 | — | |
LBGWJOVJGRVENJ
|
8.9 | IC50 | 2 | — | |
LQMGIPSONLJQKI
|
8.9 | IC50 | 2 | — | |
KYKOIMZZEJVBFT
|
8.9 | IC50 | 2 | — | |
OPKNMHGENLTFEX
|
8.9 | IC50 | 2 | — | |
AFUBZZDOEBNYBN
|
8.9 | IC50 | 2 | — | |
DTBWLHQLECJGTI
|
8.9 | IC50 | 2 | — | |
XKOPYVMSQOJAFI
|
8.9 | IC50 | 2 | — | |
DENYZIUJOTUUNY
|
8.9 | IC50 | 5 | — | |
LFYTWGBFZMCREV
|
8.9 | IC50 | 2 | — | |
PNRISLRFARDPOP
|
8.9 | IC50 | 2 | — | |
PVTGCPNFDHKZPA
|
8.9 | IC50 | 2 | — | |
SIYIOSPVPCJZFQ
|
8.9 | IC50 | 2 | — | |
AEUHXAJXFXCXEC
|
8.9 | IC50 | 2 | — | |
COFWMMMCLUXKJJ
|
8.9 | IC50 | 2 | — | |
POVQQXDQCONOIG
|
8.9 | IC50 | 2 | — | |
DKPPZBXQLWTONY
|
8.8 | IC50 | 2 | — | |
GMJHIXVSXIAXBU
|
8.8 | IC50 | 2 | — | |
QUIUMUGBDFCYNM
|
8.8 | IC50 | 2 | — | |
YNBQAYKYNYRCCA
|
8.8 | IC50 | 2 | — | |
IEJFYBWWOFTCCL
|
8.8 | IC50 | 2 | — | |
CANZSPMXSMUSHQ
|
8.8 | IC50 | 2 | — | |
CXANDIUMTJKCEI
|
8.8 | IC50 | 3 | — | |
FEAZPCVGCIRWDR
|
8.8 | IC50 | 7 | — | |
JHBYKLGSLRTFEJ
|
8.8 | IC50 | 2 | — | |
SUFCRESGNWZKKU
|
8.8 | IC50 | 2 | — | |
QTBPBWJIVQWNSL
|
8.8 | IC50 | 2 | — | |
ANAQCVXUMUTPJY
|
8.8 | IC50 | 3 | — | |
BYRSMXQNHWADRE
|
8.8 | IC50 | 2 | — | |
SQDLSZSGNSLBEQ
|
8.8 | IC50 | 2 | — | |
HMABYWSNWIZPAG
|
8.8 | IC50 | 12 | — | |
QNQFPYADHVFRKQ
|
8.8 | IC50 | 5 | — | |
URCVWNDRSBFBMR
|
8.8 | IC50 | 2 | — | |
XSNNYLLCIBEWBI
|
8.7 | IC50 | 2 | — | |
HRTOLPFSQSROQU
|
8.7 | IC50 | 2 | — | |
RJIZKFOPJCXLAT
|
8.7 | IC50 | 2 | — |