Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FVQRNLFWMRQUPL
|
9.2 | IC50 | 2 | — | |
HIQNGQBSWOVLFK
|
9.2 | IC50 | 2 | — | |
HWGQMRYQVZSGDQ
|
9.2 | IC50 | 7 | — | |
QKKMIWPBDBLRBT
|
9.2 | IC50 | 3 | — | |
QOKRGHZZWOEZGQ
|
9.2 | IC50 | 2 | — | |
SDQYXOQWRCKNII
|
9.2 | IC50 | 2 | — | |
UYSWVENMUWDLDZ
|
9.2 | IC50 | 2 | — | |
IFVPMPLYZAFFCS
|
9.2 | IC50 | 2 | — | |
KGKRAZRBCRNYFN
|
9.2 | IC50 | 2 | — | |
UXPFVYUKTWOUJT
|
9.2 | IC50 | 2 | — | |
ZBAXELGETHXFPG
|
9.2 | IC50 | 2 | — | |
OIUDYISXHDWWQJ
|
9.2 | IC50 | 2 | — | |
ORXLIHVWCSCXBW
|
9.2 | IC50 | 2 | — | |
GTCQRARQFNUVRK
|
9.2 | IC50 | 3 | — | |
JNMWDFWEHGHKSH
|
9.2 | IC50 | 2 | — | |
NUSUZBNCZDEMNE
|
9.2 | IC50 | 2 | — | |
CVEWKKYMSPEHGN
|
9.2 | IC50 | 2 | — | |
KIUHBHFVVQQALF
|
9.2 | Ki | 9 | — | |
ZSAAKXQVHMDJNL
|
9.2 | IC50 | 2 | — | |
ZTEDLCUEUUWRAT
|
9.2 | IC50 | 3 | — | |
AVOBSJNOVKNJNP
|
9.1 | IC50 | 2 | — | |
QNPIRVLIJKKNNX
|
9.1 | IC50 | 2 | — | |
UWTWKRHBLDCXHT
|
9.1 | IC50 | 2 | — | |
NSRSVDVZPFIILV
|
9.1 | IC50 | 2 | — | |
QKZGOZNDFYDQOV
|
9.1 | IC50 | 2 | — | |
XEBAVJCPTDOUIT
|
9.1 | IC50 | 2 | — | |
FWPWZSSWINQBHB
|
9.1 | IC50 | 2 | — | |
RYCVFUGCROLXMH
|
9.1 | IC50 | 2 | — | |
VGOGMUIBXGGDAR
|
9.1 | IC50 | 2 | — | |
AXXNBSKROWNMJJ
|
9.1 | IC50 | 2 | — | |
CANZSPMXSMUSHQ
|
9.1 | IC50 | 2 | — | |
IXUDDAPEXVCPBQ
|
9.1 | IC50 | 2 | — | |
PPHPURVUIFAHQD
|
9.1 | IC50 | 2 | — | |
QKZGOZNDFYDQOV
|
9.1 | IC50 | 2 | — | |
WHQIULPFILPYJQ
|
9.1 | IC50 | 2 | — | |
XCIJWZABVFOSOA
|
9.1 | IC50 | 2 | — | |
ZCZXHBMPYFPNQW
|
9.1 | IC50 | 2 | — | |
QGOJFKKLWHNNFG
|
9.0 | IC50 | 7 | — | |
OMPYCYLPJBIPKG
|
9.0 | IC50 | 2 | — | |
WKXCQZQWHUTWSY
|
9.0 | IC50 | 5 | — | |
FNXYFOFBZPBUFN
|
9.0 | IC50 | 2 | — | |
OQFPIZQVUQJWMS
|
9.0 | IC50 | 2 | — | |
CQDSSYSRDXRGLW
|
9.0 | IC50 | 2 | — | |
NBNNIAGURKGWAO
|
9.0 | IC50 | 2 | — | |
PVRVKAMGYYHFJO
|
9.0 | IC50 | 3 | — | |
AHIVQGOUBLVTCB
|
9.0 | Ki | 2 | — | |
AOLFJVDCFAXDOZ
|
9.0 | IC50 | 4 | — | |
BFJMBXAFUUTYIR
|
9.0 | IC50 | 2 | — | |
CANZSPMXSMUSHQ
|
9.0 | IC50 | 2 | — | |
NFPIZUDTGKCWQL
|
9.0 | Ki | 2 | — |