Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XQFNOSLDNBPLNW
|
6.1 | IC50 | 2 | — | |
SSRCPYMXFHISQW
|
6.1 | IC50 | 3 | — | |
ACVZUAKWEUBENM
|
6.1 | IC50 | 2 | — | |
ANAUZAZPUGQDNM
|
6.1 | IC50 | 3 | — | |
FDICCIFLUUYDFS
|
6.1 | IC50 | 4 | — | |
IFGZJOCKQVPMQP
|
6.1 | IC50 | 3 | — | |
MOMSZDNLTDTPMD
|
6.1 | IC50 | 3 | — | |
NFBXUOSSYJJKFK
|
6.1 | IC50 | 2 | — | |
WLZJEOODSSBWMB
|
6.1 | IC50 | 3 | — | |
ZVPOJSOOBYKHHV
|
6.1 | IC50 | 2 | — | |
JWTZFQHEWRUOBW
|
6.1 | IC50 | 3 | — | |
LBCRVQOCKRRJPU
|
6.1 | IC50 | 2 | — | |
LANJYZWTSUUASB
|
6.1 | IC50 | 3 | — | |
KZLPIRPQDKFMRG
|
6.1 | IC50 | 3 | — | |
YAAIOGGCMLWOPM
|
6.1 | IC50 | 4 | — | |
OIOQXLAIFONXGK
|
6.1 | IC50 | 2 | — | |
WDAVNQKSHQVPKD
|
6.1 | IC50 | 4 | — | |
CADYSKUZMAIDBU
|
6.0 | IC50 | 4 | — | |
CKOUULRCBKAWEI
|
6.0 | IC50 | 4 | — | |
HTLUBFSSIMOABR
|
6.0 | IC50 | 3 | — | |
LQJVOLSLAFIXSV
|
6.0 | IC50 | 4 | — | |
UQSSCRPZDDBPIX
|
6.0 | IC50 | 3 | — | |
FVSMOECHMBICED
|
6.0 | IC50 | 3 | — | |
WADUGMWGTNMWRD
|
6.0 | IC50 | 3 | — | |
WWNPUHZOGTUNGR
|
6.0 | IC50 | 3 | — | |
MPXAEYSGFKRDQM
|
6.0 | IC50 | 7 | — | |
QONNTUSBURAFST
|
6.0 | IC50 | 4 | — | |
DTMHAFMUJHYVGK
|
6.0 | IC50 | 3 | — | |
JDZQHCQYJAHSCQ
|
6.0 | IC50 | 3 | — | |
ZPTIGCVQFHKQDB
|
6.0 | IC50 | 3 | — | |
FNBQKJSMQWRTEK
|
6.0 | IC50 | 2 | — | |
FSNRYQUQAYKAPH
|
6.0 | IC50 | 4 | — | |
JMPCTCLDKNUTHJ
|
6.0 | IC50 | 4 | — | |
OOIMOZIUYZYXLA
|
6.0 | IC50 | 2 | — | |
YFRRHPBZXLBANM
|
6.0 | IC50 | 3 | — | |
ZJNATVSUTRSLJP
|
6.0 | IC50 | 3 | — |