Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRGTYYQXOBIJNO
|
6.4 | IC50 | 3 | — | |
AKGAPIJDXHPECB
|
6.4 | IC50 | 2 | — | |
BMZFSQDDGKZEHW
|
6.4 | IC50 | 3 | — | |
QPPRMYWGJMMFHW
|
6.4 | IC50 | 2 | — | |
LVTXKTNJLIESPY
|
6.4 | IC50 | 2 | — | |
UTEHUKGJDLVHIH
|
6.4 | IC50 | 3 | — | |
HANJAZOKICPNAX
|
6.4 | IC50 | 3 | — | |
QEZFXBJCFJZWMT
|
6.4 | IC50 | 2 | — | |
ZJHLKLRWORVGKO
|
6.4 | IC50 | 3 | — | |
BPRGXQTYABGOBA
|
6.3 | IC50 | 3 | — | |
AFHDZWZQZNOEPI
|
6.3 | IC50 | 4 | — | |
FCOPXWHSTOLCAJ
|
6.3 | IC50 | 2 | — | |
JZKVDRXHUJSBJE
|
6.3 | IC50 | 2 | — | |
ZAVBKFISCRSHAT
|
6.3 | IC50 | 2 | — | |
ZFGIVIZXCYOWBK
|
6.3 | IC50 | 16 | — | |
BANSZVBMEHYKAV
|
6.3 | IC50 | 4 | — | |
WHHFINHFBVESNP
|
6.3 | IC50 | 2 | — | |
DKPIHFWBNZVINS
|
6.3 | IC50 | 2 | — | |
PTKGBRUVUGNNDZ
|
6.3 | IC50 | 2 | — | |
RFMIZKCQNUDSTO
|
6.3 | IC50 | 3 | — | |
UORYBBKJEVGLPQ
|
6.3 | IC50 | 2 | — | |
XFDGHNYVTUXZDC
|
6.3 | IC50 | 2 | — | |
IZGNMSCICRBUAB
|
6.3 | IC50 | 3 | — | |
VHNNUIFUWOPIHC
|
6.3 | IC50 | 2 | — | |
MCCQXQRJNJXHRG
|
6.2 | IC50 | 3 | — | |
QZHUFUOXNJRYML
|
6.2 | IC50 | 4 | — | |
UOHKZMQXEJGUES
|
6.2 | IC50 | 4 | — | |
IWIXTZQBCXYDRG
|
6.2 | IC50 | 3 | — | |
WQGFJZQGDWKRMN
|
6.2 | IC50 | 4 | — | |
AOMPHWKJTUPEOB
|
6.2 | IC50 | 3 | — | |
IESAQQWECFSSTH
|
6.2 | IC50 | 2 | — | |
XTEDLLOZIRDMGM
|
6.2 | IC50 | 3 | — | |
MGEFDMCHHLACOB
|
6.2 | IC50 | 4 | — | |
NGWLKFVMSQZGRO
|
6.2 | IC50 | 3 | — | |
OAXRVCSFISVGCI
|
6.2 | IC50 | 3 | — | |
RGSSADMOZOOPCT
|
6.2 | IC50 | 4 | — | |
FSJBONLMIKLDFZ
|
6.2 | IC50 | 2 | — | |
QWKZXCNQEFMJAM
|
6.2 | IC50 | 3 | — | |
RDAGLFLFHKNHGG
|
6.2 | IC50 | 2 | — | |
NJLMHMDGCCRWFC
|
6.2 | IC50 | 2 | — | |
OUYAJDGIWDVAJZ
|
6.2 | IC50 | 2 | — | |
VSWDXFSNRCBKQK
|
6.2 | IC50 | 2 | — | |
YAARIUWCZZVAFB
|
6.2 | IC50 | 2 | — | |
JCFJQIHDZHHMQT
|
6.2 | Ki | 42 | — | |
VJHDAFXRSRJKPL
|
6.2 | IC50 | 3 | — | |
VKQCBCMAFAIWOE
|
6.2 | IC50 | 3 | — | |
FHBYLOWAINBPRJ
|
6.2 | IC50 | 4 | — | |
CSZYQIKNQBWYMC
|
6.1 | IC50 | 3 | — | |
OEHCCJHWIUUHFU
|
6.1 | IC50 | 3 | — | |
AOMPHWKJTUPEOB
|
6.1 | IC50 | 3 | — |