Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HLOAWTDOVMWWAG
|
6.7 | IC50 | 2 | — | |
KNAIHOJCNBJITI
|
6.7 | IC50 | 3 | — | |
YFUQBDLMKVLYPM
|
6.7 | IC50 | 20 | — | |
YTQLCJYUTMBQFF
|
6.7 | IC50 | 2 | — | |
BLVQSAHMDXWBNC
|
6.7 | IC50 | 2 | — | |
GGQAXNFSEUSJJE
|
6.7 | IC50 | 3 | — | |
OWLIGWULYLQYLA
|
6.7 | IC50 | 2 | — | |
UYFDUBXEDXZHBG
|
6.7 | IC50 | 2 | — | |
IPPGXRJXMXVNLN
|
6.6 | IC50 | 3 | — | |
IYJYZOJIOGICFK
|
6.6 | IC50 | 2 | — | |
QHKQUHOWXBJVAF
|
6.6 | IC50 | 2 | — | |
MDURPWFKFWBOHZ
|
6.6 | IC50 | 2 | — | |
AVTNDVTVXDIHDQ
|
6.6 | IC50 | 2 | — | |
WHPSHUGOCRYIEA
|
6.6 | IC50 | 20 | — | |
SEFVDSHLUATZOI
|
6.6 | IC50 | 2 | — | |
FHWNIOZFSDHKSG
|
6.6 | IC50 | 4 | — | |
VEVDSJNRSJPWSK
|
6.6 | IC50 | 2 | — | |
NXRCVVIFMJBFPF
|
6.6 | IC50 | 3 | — | |
TWAKELMLSWVDPB
|
6.6 | IC50 | 2 | — | |
AUNVTZZLENFGSL
|
6.6 | IC50 | 2 | — | |
HIDGSHNRMYFZHS
|
6.6 | IC50 | 2 | — | |
SOWWGFRAFDIXID
|
6.6 | IC50 | 20 | — | |
YPLLSXUOZDMWPL
|
6.5 | IC50 | 2 | — | |
FNYTYXJFOSRUTI
|
6.5 | IC50 | 3 | — | |
HETSSARHFAGODR
|
6.5 | IC50 | 3 | — | |
IGFFHJGCUWZRKD
|
6.5 | IC50 | 20 | — | |
QWXXAMNXENCFLM
|
6.5 | IC50 | 2 | — | |
BCSYLIBZTSVMJI
|
6.5 | IC50 | 3 | — | |
ZYPRPLRGMSHRRW
|
6.5 | IC50 | 2 | — | |
GVMXJRXJKMOCBF
|
6.5 | IC50 | 2 | — | |
UIPJAQKAZCQVPU
|
6.5 | IC50 | 3 | — | |
CXHGLEPFSZKWBR
|
6.5 | IC50 | 2 | — | |
KXIWZPLTJFWCLG
|
6.5 | IC50 | 2 | — | |
SSRCPYMXFHISQW
|
6.5 | IC50 | 3 | — | |
UEEAPWCOJZPFBY
|
6.5 | IC50 | 2 | — | |
DIXJAUCKOHDBNI
|
6.5 | IC50 | 2 | — | |
HBRPUCMYDQNVOS
|
6.5 | IC50 | 3 | — | |
HDXNXKLFFUORPE
|
6.5 | IC50 | 2 | — | |
JXORYUCIOICGOX
|
6.5 | IC50 | 3 | — | |
PYZXOAIEYXKOIA
|
6.5 | IC50 | 2 | — | |
RMTXPZAKIDWSDV
|
6.5 | IC50 | 2 | — | |
RZFVLEJOHSLEFR
|
6.5 | IC50 | 4 | — | |
RTVLFJXYETXJBN
|
6.5 | IC50 | 2 | — | |
XMNISQQDQQVTBJ
|
6.5 | IC50 | 4 | — | |
FMSBJUGTJUGWQX
|
6.4 | IC50 | 2 | — | |
IJTBFOMRKCFLIG
|
6.4 | IC50 | 2 | — | |
AXVJLHNEUCXOHA
|
6.4 | IC50 | 2 | — | |
ZQAMFUHPGNZLHA
|
6.4 | IC50 | 3 | — | |
JKUCQWSEJQYAJC
|
6.4 | IC50 | 3 | — | |
BCSYLIBZTSVMJI
|
6.4 | IC50 | 3 | — |