Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OSSMVMKSVHUBNI
|
7.2 | IC50 | 2 | — | |
JGLLGSHEXZAGLB
|
7.2 | IC50 | 2 | — | |
MEPVROYUXYYJJC
|
7.2 | IC50 | 2 | — | |
UHBZXJKZJXSEBM
|
7.2 | IC50 | 2 | — | |
CPGPHRFTIHQLET
|
7.2 | IC50 | 2 | — | |
LXCLGXFJSUMMJY
|
7.2 | IC50 | 4 | — | |
RGOOUZDKFUXEGZ
|
7.2 | IC50 | 2 | — | |
IQDRXCXNISQMPH
|
7.2 | IC50 | 3 | — | |
BTXUKBPFPHAMAC
|
7.2 | IC50 | 2 | — | |
QHEYBDYWUSNRBP
|
7.1 | IC50 | 2 | — | |
HSICEIFWMLSUPK
|
7.1 | IC50 | 2 | — | |
LCKFRXLDDGHRAM
|
7.1 | IC50 | 2 | — | |
MSOMGRYOZBJWOT
|
7.1 | Kd | 2 | — | |
WTZXJCZLEYCTSS
|
7.1 | IC50 | 2 | — | |
GWBSSUZALYDTAX
|
7.1 | IC50 | 3 | — | |
HISJVPLDLOXJOH
|
7.1 | IC50 | 2 | — | |
QLQTUEDKHBEEJG
|
7.1 | IC50 | 2 | — | |
AYBCRDPWFPGRPP
|
7.1 | IC50 | 2 | — | |
BIFMDHUVYGGFCU
|
7.1 | IC50 | 10 | — | |
IBWYFZTUWYBKBG
|
7.1 | IC50 | 2 | — | |
IPJVKKPTQCQECT
|
7.1 | Kd | 2 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
OVXXLTCZEHZISR
|
7.1 | IC50 | 2 | — | |
RMPXVEDDRZOQIA
|
7.1 | IC50 | 2 | — | |
HNVGNPZHTCPRJL
|
7.1 | IC50 | 2 | — | |
VOQLJAINULFPEC
|
7.1 | IC50 | 2 | — | |
AUSDJKWCUGOMRT
|
7.1 | IC50 | 2 | — | |
BMXUSXFYGFJVNI
|
7.1 | IC50 | 2 | — | |
VARCSQSOWLMGTH
|
7.1 | Kd | 2 | — | |
BSJKOBUSZMTFLW
|
7.0 | IC50 | 2 | — | |
HGBGVYVWYQKXTN
|
7.0 | Kd | 2 | — | |
RHCZTJJJLXGIDT
|
7.0 | IC50 | 4 | — | |
INOWNSTVYAHHRD
|
7.0 | IC50 | 2 | — | |
ONYDOUQLFUMDET
|
7.0 | IC50 | 2 | — | |
RVOUDNBEIXGHJY
|
7.0 | IC50 | 2 | — | |
BSBYIGMCJVUHQV
|
7.0 | IC50 | 2 | — | |
RUOPPILAFNBOIX
|
7.0 | IC50 | 2 | — | |
FELISMCMXIVCLT
|
7.0 | IC50 | 2 | — | |
PPLKPFGRKQMGRE
|
7.0 | IC50 | 3 | — | |
ATXBWTLLRQPRTF
|
7.0 | IC50 | 20 | — | |
XKPGTGFSIKPAND
|
7.0 | IC50 | 20 | — | |
CRLANDXFFHDDAK
|
7.0 | IC50 | 20 | — | |
JKXYPJZBOPXUBC
|
7.0 | IC50 | 2 | — | |
JNLILESBBKKTIC
|
7.0 | IC50 | 2 | — | |
KAPAUCQOBGHPCQ
|
7.0 | IC50 | 2 | — | |
WCZAODKSIJSHQD
|
7.0 | IC50 | 2 | — | |
WMCXYGMSZGSRSX
|
7.0 | IC50 | 2 | — | |
YMRLPMGPWVJHRW
|
7.0 | IC50 | 20 | — | |
ZUWRJCHNQXZPKT
|
7.0 | IC50 | 2 | — | |
AUGRKZAFBVCEBZ
|
7.0 | IC50 | 2 | — |