Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ANXZOJPKYNUICG
|
7.4 | IC50 | 2 | — | |
CEJMJSUDCBTVDD
|
7.4 | IC50 | 2 | — | |
LZKGLICEGUTSDW
|
7.4 | IC50 | 3 | — | |
NUHZJIJDJJVSKK
|
7.4 | IC50 | 3 | — | |
ZZFIQKPNOYYXIV
|
7.4 | IC50 | 2 | — | |
KRLQJSZEXYIYPQ
|
7.4 | IC50 | 2 | — | |
IADDRMVOCUHETH
|
7.4 | IC50 | 2 | — | |
INLBHAOCYUPABD
|
7.4 | IC50 | 2 | — | |
NBVFKEHFDGGDFT
|
7.4 | IC50 | 2 | — | |
YUVLMYMBEWNHPA
|
7.4 | IC50 | 2 | — | |
KTIYJXKGHKLGEV
|
7.4 | IC50 | 3 | — | |
LAKYTXYAGBFERQ
|
7.4 | IC50 | 2 | — | |
NALBIBKGPRRCCO
|
7.4 | IC50 | 2 | — | |
VVVYIXNVAPSYSE
|
7.4 | IC50 | 3 | — | |
DDFLFKTXUWPNMV
|
7.3 | IC50 | 3 | — | |
DDFLFKTXUWPNMV
|
7.3 | IC50 | 3 | — | |
KKRQGICUYMCZFH
|
7.3 | IC50 | 2 | — | |
GNEBUQTZKVXTKB
|
7.3 | IC50 | 2 | — | |
OKZVWHVKFPRNLX
|
7.3 | IC50 | 2 | — | |
WEVHGUILVANSPZ
|
7.3 | IC50 | 2 | — | |
NDFQKILREVNCLZ
|
7.3 | IC50 | 2 | — | |
PGGOMVDSVVGTHN
|
7.3 | IC50 | 2 | — | |
SAJUIWASIJXNSM
|
7.3 | IC50 | 2 | — | |
SAJUIWASIJXNSM
|
7.3 | IC50 | 2 | — | |
UEGWFDZLXJTQDG
|
7.3 | IC50 | 2 | — | |
UNIBAROCFQUNJP
|
7.3 | IC50 | 2 | — | |
XURWTHPKVQLLQP
|
7.3 | Kd | 2 | — | |
HICODDHJHKXOBW
|
7.3 | IC50 | 2 | — | |
JHEWPSFLMCUPRO
|
7.3 | IC50 | 2 | — | |
LXMVOWGBBQUTCO
|
7.3 | IC50 | 2 | — | |
ADRLWUFSRZSWAB
|
7.3 | IC50 | 2 | — | |
NHTFNTYBBURGHS
|
7.3 | IC50 | 2 | — | |
NLWYFXIKIPVWHJ
|
7.3 | IC50 | 2 | — | |
QFKIZAYSXMBONY
|
7.3 | IC50 | 2 | — | |
KDPQFXRDUUVUMM
|
7.3 | IC50 | 2 | — | |
FITDTEZFVLDGBX
|
7.3 | IC50 | 2 | — | |
PTRXVEZPOQLFDC
|
7.3 | IC50 | 2 | — | |
QYFRQINXIBOIOI
|
7.3 | IC50 | 2 | — | |
UEGWFDZLXJTQDG
|
7.3 | IC50 | 2 | — | |
HTBJXITVMAAPGH
|
7.2 | IC50 | 2 | — | |
NKJYUBWSGJMPAJ
|
7.2 | IC50 | 2 | — | |
WGTJWDKKJAQXMI
|
7.2 | Kd | 2 | — | |
WQVZBZQCVBIXLT
|
7.2 | IC50 | 3 | — | |
AROUQFRRWYAJHE
|
7.2 | IC50 | 2 | — | |
BDQLEBFPVSEZSI
|
7.2 | IC50 | 2 | — | |
GNPXWZUQWUCREF
|
7.2 | Kd | 2 | — | |
KCCHUDANIWRWFS
|
7.2 | IC50 | 3 | — | |
TXIZSRVUVVGWCN
|
7.2 | IC50 | 2 | — | |
CHRQYHKDXOIBPC
|
7.2 | IC50 | 2 | — | |
DCYHJVFMNYSPNT
|
7.2 | IC50 | 9 | — |