Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CHUANYXVPMSWFM
|
7.6 | IC50 | 3 | — | |
HEDHFDLLWZBOLO
|
7.6 | IC50 | 2 | — | |
JJCAYWVTBMMQMQ
|
7.6 | IC50 | 2 | — | |
LHXVNDXPHWSUGM
|
7.6 | IC50 | 2 | — | |
LWYGAYYSBCIGHJ
|
7.6 | Ki | 2 | — | |
MJCWPISTEYQNBA
|
7.6 | IC50 | 2 | — | |
RSFVVMOORBEYQG
|
7.6 | IC50 | 2 | — | |
RVBDGUXYQPDTTD
|
7.6 | IC50 | 2 | — | |
UBMGXAJVWWFLCY
|
7.6 | IC50 | 2 | — | |
XCMZWTDSYWVLET
|
7.6 | IC50 | 2 | — | |
AXAVOVXYAFPCSL
|
7.6 | IC50 | 2 | — | |
USANDOAEVNQHRL
|
7.6 | IC50 | 2 | — | |
MKRASBLHKPMOJK
|
7.5 | IC50 | 20 | — | |
QBGORSWTCHSEMS
|
7.5 | IC50 | 2 | — | |
YFRJWFALOKTWJY
|
7.5 | IC50 | 3 | — | |
SAVQIVUHYCZXGH
|
7.5 | IC50 | 2 | — | |
UBMGXAJVWWFLCY
|
7.5 | IC50 | 2 | — | |
OWJIPVZWQPNFLC
|
7.5 | IC50 | 2 | — | |
KTIYJXKGHKLGEV
|
7.5 | IC50 | 3 | — | |
MABHSRSWSCMJOM
|
7.5 | IC50 | 2 | — | |
PXVGNWOIQRDFEX
|
7.5 | IC50 | 2 | — | |
UNJCZSCIWNQLFD
|
7.5 | IC50 | 2 | — | |
URLKBSWMVHJNHY
|
7.5 | IC50 | 2 | — | |
USTBPCWKZJLWHI
|
7.5 | IC50 | 2 | — | |
DOKFTMCJGVGNMI
|
7.5 | IC50 | 2 | — | |
LTUOFKFLZDKSRD
|
7.5 | IC50 | 2 | — | |
QMFJNBILTNXCGW
|
7.5 | Kd | 2 | — | |
WUSATWKNDGXYRU
|
7.5 | IC50 | 2 | — | |
WOBDQRLNYWLLJQ
|
7.5 | IC50 | 2 | — | |
CXHHTZQIOFCSNN
|
7.5 | IC50 | 2 | — | |
HBJRTNJBCUCSST
|
7.5 | IC50 | 2 | — | |
JGWQDYTVDJMRNI
|
7.5 | Kd | 2 | — | |
QYXDDRWHQGGYKR
|
7.5 | IC50 | 2 | — | |
DNTOQLUATWVLNE
|
7.5 | IC50 | 2 | — | |
VQUQBABVYFSBGV
|
7.5 | IC50 | 6 | — | |
CQDSSYSRDXRGLW
|
7.4 | IC50 | 2 | — | |
FCXORJBFYRYCGS
|
7.4 | IC50 | 2 | — | |
HICODDHJHKXOBW
|
7.4 | IC50 | 2 | — | |
UEGWFDZLXJTQDG
|
7.4 | IC50 | 2 | — | |
UJTLXFAELPEGKX
|
7.4 | IC50 | 2 | — | |
UNPLREWLHBUEMG
|
7.4 | IC50 | 2 | — | |
XNYVULHMPZSVEK
|
7.4 | IC50 | 2 | — | |
AJCFYLHZMCTQJH
|
7.4 | IC50 | 3 | — | |
DFLMYYBQQIIOLC
|
7.4 | IC50 | 2 | — | |
FMVGMOVFNFTMQG
|
7.4 | IC50 | 2 | — | |
KQRUVCRIBJGRNK
|
7.4 | IC50 | 2 | — | |
UQZCQKXJAXKZQH
|
7.4 | IC50 | 4 | — | |
QTAAMFZROWGTBV
|
7.4 | IC50 | 2 | — | |
UZPYETATKJIYAI
|
7.4 | IC50 | 2 | — | |
XKBLRQOXNMSXTO
|
7.4 | IC50 | 2 | — |