Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CQDSSYSRDXRGLW
|
7.8 | IC50 | 2 | — | |
HLAHINFHXDROJP
|
7.8 | IC50 | 2 | — | |
HPNPGKDJVPSETA
|
7.8 | IC50 | 2 | — | |
IOHRTULIGFHGAL
|
7.8 | Ki | 2 | — | |
KQURMMMJBDYUSN
|
7.8 | IC50 | 2 | — | |
KYZJKYGUVGFTFT
|
7.8 | IC50 | 2 | — | |
WJSBPAZKQYZPAE
|
7.8 | IC50 | 2 | — | |
TXIZSRVUVVGWCN
|
7.8 | IC50 | 2 | — | |
RBANKGXIRGNBSA
|
7.8 | IC50 | 2 | — | |
SBJGLDKVXLKVPI
|
7.8 | IC50 | 2 | — | |
QJULBGPNAODEGM
|
7.8 | IC50 | 2 | — | |
UVYVRAATXCFMQQ
|
7.8 | IC50 | 4 | — | |
UWPDADPDWVTOEC
|
7.8 | IC50 | 2 | — | |
DXFARVNRLJXDDA
|
7.7 | IC50 | 2 | — | |
MHEGXLWYODUJMQ
|
7.7 | IC50 | 2 | — | |
MJPLTIGFNFYZIV
|
7.7 | IC50 | 2 | — | |
DAIMOGAYMHVUBZ
|
7.7 | IC50 | 2 | — | |
AFVMAFOLQJXDAD
|
7.7 | IC50 | 2 | — | |
LVZZNRAHJDTKAL
|
7.7 | IC50 | 2 | — | |
NBNNIAGURKGWAO
|
7.7 | IC50 | 2 | — | |
OTDIMNJLKVGGOB
|
7.7 | IC50 | 3 | — | |
CTLOSZHDGZLOQE
|
7.7 | IC50 | 2 | — | |
FUUOPLKUAWRLLD
|
7.7 | IC50 | 2 | — | |
KHGMRXFPRSSDPX
|
7.7 | IC50 | 2 | — | |
OOMGICXJISMCLR
|
7.7 | IC50 | 2 | — | |
POAFYPSDLXGQBX
|
7.7 | IC50 | 3 | — | |
URLKBSWMVHJNHY
|
7.7 | IC50 | 2 | — | |
WPZCNAVAWRYPHY
|
7.7 | IC50 | 4 | — | |
YMBFFLHVYTXNDP
|
7.7 | IC50 | 2 | — | |
OTEFEZRIUOWLMH
|
7.7 | IC50 | 2 | — | |
GYUCFGYTWSIWKA
|
7.7 | IC50 | 2 | — | |
WJSBPAZKQYZPAE
|
7.7 | IC50 | 2 | — | |
YNOAURUBJUTHDB
|
7.7 | IC50 | 2 | — | |
ZANJWUNZMOCQFD
|
7.7 | IC50 | 2 | — | |
BPWNUTSKZNJOAK
|
7.7 | IC50 | 2 | — | |
OYGLTKXMFGWXJT
|
7.7 | IC50 | 2 | — | |
VAXCTJXSWDBQDO
|
7.6 | IC50 | 2 | — | |
FZWPUFVVEGJNEV
|
7.6 | IC50 | 2 | — | |
IMVSOTHSTUMFCM
|
7.6 | IC50 | 2 | — | |
MWLJLVHPVHBVDL
|
7.6 | IC50 | 3 | — | |
BVEJDOKUOZXSCO
|
7.6 | IC50 | 2 | — | |
CBRIZHZYFLCPAP
|
7.6 | IC50 | 3 | — | |
IRUQIRGVTCDGBO
|
7.6 | IC50 | 2 | — | |
PNPZDTYSNSOILZ
|
7.6 | IC50 | 2 | — | |
SLIPNSLITDGVIT
|
7.6 | IC50 | 2 | — | |
SOKIJBHBGDDEGH
|
7.6 | IC50 | 2 | — | |
TZJJVUZBPNABSN
|
7.6 | IC50 | 2 | — | |
VRLLUDPWEDVARZ
|
7.6 | IC50 | 2 | — | |
IRXHYIYBIYVZMS
|
7.6 | IC50 | 2 | — | |
XPKUFZAKPWQMOR
|
7.6 | IC50 | 2 | — |