Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XDVDXJJYSVRAJX
|
8.0 | IC50 | 2 | — | |
XFINPBQKFDIRJH
|
8.0 | IC50 | 3 | — | |
RRTBNWLSPAIIKM
|
7.9 | IC50 | 2 | — | |
YADMFPWTDIQDHU
|
7.9 | IC50 | 2 | — | |
JJDFDZDTXGPNIC
|
7.9 | IC50 | 2 | — | |
WEKCQPVMVKJTQD
|
7.9 | IC50 | 2 | — | |
DRLOBUZZJYWFDE
|
7.9 | IC50 | 2 | — | |
DUFXFZVTFQWSQI
|
7.9 | IC50 | 2 | — | |
FWZKUFCCKVNCSL
|
7.9 | IC50 | 2 | — | |
IEFSYHDGPQTMNE
|
7.9 | IC50 | 2 | — | |
MUUFHIOSFYMTJG
|
7.9 | IC50 | 2 | — | |
QTONZRQJLGKQRC
|
7.9 | Ki | 2 | — | |
RPIXUTROJMVGDZ
|
7.9 | IC50 | 2 | — | |
MWLJLVHPVHBVDL
|
7.9 | IC50 | 2 | — | |
UWIOUEAALWYOMW
|
7.9 | IC50 | 3 | — | |
HWGQMRYQVZSGDQ
|
7.9 | IC50 | 6 | — | |
RQIZHRJCWXOIGA
|
7.9 | IC50 | 2 | — | |
ACCULLWIBRVLMN
|
7.9 | IC50 | 2 | — | |
HDFQNQPMGAHQTL
|
7.9 | IC50 | 5 | — | |
PVIVFFQABAVRDM
|
7.9 | IC50 | 2 | — | |
WFZXKJNCDQJJDD
|
7.9 | IC50 | 2 | — | |
MSZHRPFWZYCRHL
|
7.9 | IC50 | 2 | — | |
ZKLQWWOVTJLLRS
|
7.9 | IC50 | 2 | — | |
MJPLTIGFNFYZIV
|
7.9 | IC50 | 2 | — | |
DFAIABHDMOLQDA
|
7.9 | IC50 | 5 | — | |
FZWPUFVVEGJNEV
|
7.9 | IC50 | 2 | — | |
OTEFEZRIUOWLMH
|
7.9 | IC50 | 2 | — | |
ZDQAOBPLFLTAOZ
|
7.9 | IC50 | 2 | — | |
CDDMAJJEUDLCTJ
|
7.8 | IC50 | 2 | — | |
CQANUCNRTBYOHB
|
7.8 | IC50 | 2 | — | |
GDUDWHVXWZWKMX
|
7.8 | IC50 | 2 | — | |
GVBZXJBCNDEVRT
|
7.8 | IC50 | 2 | — | |
KORBVNCZCNDJHA
|
7.8 | IC50 | 2 | — | |
NPOFZKXRQDDDDY
|
7.8 | IC50 | 2 | — | |
OWOZSIHFAFXWTN
|
7.8 | IC50 | 2 | — | |
RLWLFXINNNSDCN
|
7.8 | IC50 | 2 | — | |
USANDOAEVNQHRL
|
7.8 | IC50 | 2 | — | |
USTBPCWKZJLWHI
|
7.8 | IC50 | 2 | — | |
VYUKSMNSIRGBBM
|
7.8 | IC50 | 2 | — | |
DETVQHYFSHWWBS
|
7.8 | IC50 | 2 | — | |
IMVSOTHSTUMFCM
|
7.8 | IC50 | 2 | — | |
OORVLKKZQATWIA
|
7.8 | IC50 | 2 | — | |
CEABYCITKOLZEE
|
7.8 | IC50 | 4 | — | |
CHXQYSSALOBPEV
|
7.8 | IC50 | 2 | — | |
HROJOEXOVRGYRB
|
7.8 | IC50 | 2 | — | |
INOWNSTVYAHHRD
|
7.8 | IC50 | 2 | — | |
PQXUCBRUEQVEIZ
|
7.8 | IC50 | 3 | — | |
WHEDMAICUFWICE
|
7.8 | IC50 | 2 | — | |
YUZWVHGUAQAWSV
|
7.8 | IC50 | 2 | — | |
NANHPXHADBZWEH
|
7.8 | IC50 | 2 | — |