Target Details
| UniProt AC | P09874 |
|---|---|
| Gene Symbol | PARP1 |
| Protein Name | Poly [ADP-ribose] polymerase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF21728 (PADR1_N) PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) PF00645 (zf-PARP) PF08063 (Zn_ribbon_PADR1) |
Summary
- Multi-target molecules 886
- Clinical molecules 0
- Avg pChEMBL 7.83
KEGG Pathways (5)
Active Molecules (886)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FOWUOSHNILCZNQ
|
10.7 | IC50 | 5 | — | |
IKWXNXBFSIAXJW
|
9.9 | IC50 | 2 | — | |
MVLQBTNVYGLHLJ
|
9.9 | IC50 | 2 | — | |
GOFREDILGIHSQV
|
9.8 | IC50 | 2 | — | |
XTRXSBQKMQIRBT
|
9.8 | IC50 | 2 | — | |
LNQNBQNAFCUCKL
|
9.8 | IC50 | 2 | — | |
KYPCNLJQBLPDKY
|
9.7 | IC50 | 2 | — | |
CKQIWMZDFHAWQD
|
9.7 | IC50 | 2 | — | |
HCNQBHIZMIYRNP
|
9.6 | IC50 | 2 | — | |
VERAONOTUBOPNI
|
9.6 | IC50 | 2 | — | |
CDZVKEJUOKVZRK
|
9.6 | IC50 | 2 | — | |
PMIVWECZXHTRTB
|
9.6 | IC50 | 2 | — | |
HZWMZRPCQMLTNS
|
9.6 | IC50 | 2 | — | |
JLVRTMBMCWYGAL
|
9.6 | IC50 | 7 | — | |
VYGPONYCLGMRIN
|
9.6 | IC50 | 2 | — | |
FGYVNBTVFXTPDO
|
9.6 | IC50 | 2 | — | |
CVEWKKYMSPEHGN
|
9.5 | IC50 | 2 | — | |
NVELEVIIIBFNQK
|
9.5 | IC50 | 2 | — | |
TZXPRLCNBIYCJF
|
9.5 | IC50 | 2 | — | |
LWIZMEPNSZKHGD
|
9.5 | IC50 | 3 | — | |
JQJWUJKFLKIJHP
|
9.5 | IC50 | 2 | — | |
NRAWTIJOODMZGX
|
9.5 | IC50 | 3 | — | |
YUBJOUADCHZSHS
|
9.5 | IC50 | 3 | — | |
WVUVFMVGYOVQEF
|
9.5 | IC50 | 2 | — | |
ACJDTAHNIFCCHB
|
9.4 | IC50 | 3 | — | |
CLTQHSPVFLJRRV
|
9.4 | IC50 | 2 | — | |
UAXBMDKETCJNCZ
|
9.4 | IC50 | 2 | — | |
VONMSJQAKXAFNE
|
9.4 | IC50 | 2 | — | |
GCONNFIRFPGVSS
|
9.4 | IC50 | 2 | — | |
GCYAKZZBZIDGIO
|
9.4 | IC50 | 2 | — | |
QNJVMKQCYBBEMX
|
9.4 | IC50 | 2 | — | |
YLCGFZJPUPHSLL
|
9.4 | IC50 | 2 | — | |
QBECCWNXJQTRHP
|
9.4 | IC50 | 2 | — | |
BIPYPQGWHHULTF
|
9.3 | IC50 | 2 | — | |
KFGBYSPMOSRKQE
|
9.3 | IC50 | 2 | — | |
OCMBSADNDFCQMF
|
9.3 | IC50 | 2 | — | |
VKONWDRHMRHORV
|
9.3 | IC50 | 2 | — | |
HBJRTNJBCUCSST
|
9.3 | IC50 | 2 | — | |
PBOOUBWKFXDCRA
|
9.3 | IC50 | 3 | — | |
XSPSNGRGTPWRHB
|
9.3 | IC50 | 3 | — | |
LSFVDOIBSNWJCD
|
9.3 | IC50 | 2 | — | |
MILZLJCTDLMQGC
|
9.3 | IC50 | 2 | — | |
PPHPURVUIFAHQD
|
9.3 | IC50 | 2 | — | |
SISUHZJVRZOQES
|
9.3 | IC50 | 2 | — | |
TZXPRLCNBIYCJF
|
9.3 | IC50 | 2 | — | |
UMBRPUOTHIKKFW
|
9.3 | IC50 | 2 | — | |
UAXBMDKETCJNCZ
|
9.3 | IC50 | 2 | — | |
UDFQFCRUNLBZKM
|
9.2 | IC50 | 3 | — | |
CANZSPMXSMUSHQ
|
9.2 | IC50 | 2 | — | |
DQFNQJDEGHPCEJ
|
9.2 | IC50 | 2 | — |