Target Details
| UniProt AC | P09871 |
|---|---|
| Gene Symbol | C1S |
| Protein Name | Complement C1s subcomponent |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00431 (CUB) PF14670 (FXa_inhibition) PF00084 (Sushi) PF00089 (Trypsin) |
Summary
- Multi-target molecules 27
- Clinical molecules 0
- Avg pChEMBL 6.47
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTGQTQBPQCRNRG
|
8.8 | IC50 | 2 | — | |
VVGBUDHDUBJJKT
|
8.0 | Ki | 2 | — | |
MQQNFDZXWVTQEH
|
7.2 | IC50 | 11 | — | |
QQRQFIXRVWJLNT
|
7.2 | IC50 | 10 | — | |
BCSYIGQLBKEYFG
|
7.2 | Ki | 4 | — | |
QXVGJSQBMXLJEN
|
6.8 | IC50 | 2 | — | |
VUWARVVMIAAMOY
|
6.4 | IC50 | 3 | — | |
VLUCTQXBQVXUNP
|
6.4 | Ki | 2 | — | |
OMMIMDGHTTXEFT
|
6.4 | Ki | 2 | — | |
QHGDTGBHXYZJHD
|
6.3 | Ki | 2 | — | |
HFUGBKCICWUZIJ
|
6.3 | Ki | 3 | — | |
CKYREKXNBZFCFF
|
6.3 | Ki | 2 | — | |
WFUWFCPVIJPOGN
|
6.3 | Ki | 2 | — | |
HZNLMAXGKJQXSL
|
6.2 | Ki | 2 | — | |
OUPJOWDHCXNNFZ
|
6.2 | Ki | 2 | — | |
PYBQUZRFYXFVJH
|
6.2 | Ki | 2 | — | |
DMRSHSWYVATHJS
|
6.1 | Ki | 2 | — | |
GKBXJOCPZBRUIG
|
6.1 | IC50 | 4 | — | |
KIGJPKCRBSBFNE
|
6.1 | Ki | 2 | — | |
VPNNTFDQKJOHAQ
|
6.1 | Ki | 2 | — | |
GVDWENUEEMSFBD
|
6.1 | Ki | 2 | — | |
WAZLNMJDGBJWQY
|
6.1 | IC50 | 2 | — | |
FLKQFRKNGNJBNP
|
6.0 | Ki | 2 | — | |
MMWKNNJFQJAFDL
|
6.0 | IC50 | 2 | — | |
QOLOIIDNXILJRE
|
6.0 | IC50 | 4 | — | |
MEKFQRDWXPJRHC
|
6.0 | Ki | 2 | — | |
IHVADESBZZCEJN
|
6.0 | Ki | 2 | — |